SCHEMBL11273015

SCHEMBL11273015

CCCCCc1nc(Cl)cc(NCCO)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.54
CYP2C19 P33261 1/20 0.54
KMT2A Q03164 2/20 0.48
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
ALDH1A1 P00352 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CDC7 O00311 1/20 0.36
ROCK2 O75116 1/20 0.36
MAP4K4 O95819 1/20 0.36
PIM1 P11309 1/20 0.36
PRKACA P17612 1/20 0.36
CDK2 P24941 1/20 0.36
GSK3B P49841 1/20 0.36
HIPK2 Q9H2X6 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
SLC29A1 Q99808 1/20 0.36
TLR8 Q9NR97 1/20 0.36
ALOX5 P09917 1/20 0.36
HRH4 Q9H3N8 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11278078 0.83 CYP2D6 (0.61) CYP2D6CYP2C19KMT2AALDH1A1SMN1; SMN2
SCHEMBL3806604 0.78 KCNH2 (0.41) KMT2ATLR8MEN1
SCHEMBL8385253 0.76 KCNH2 (0.44) ESR1ALDH1A1
SCHEMBL9380817 0.75 ESR1 (0.34) KMT2AESR1ESR2SMN1; SMN2MEN1
SCHEMBL305259 0.73 CYP2D6 (0.65) CYP2D6CYP2C19KMT2AALDH1A1SMN1; SMN2
SCHEMBL9217028 0.73 CYP2D6 (0.69) CYP2D6CYP2C19KMT2AESR1ALDH1A1
SCHEMBL2578650 0.72 KMT2A (0.47) CYP2D6CYP2C19KMT2AESR1ESR2
SCHEMBL1321965 0.72 KMT2A (0.39) KMT2AESR1ESR2ALDH1A1TLR8
SCHEMBL13329883 0.72 DNM2 (0.57) ESR1ESR2ALDH1A1SMN1; SMN2TLR8
SCHEMBL13329881 0.72 DNM2 (0.57) ESR1ESR2ALDH1A1SMN1; SMN2TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0004173-B1 2,3-DIHYDROIMIDAZO (1,2-C) PYRIMIDINES, THEIR PREPARATION, FORMULATIONS CONTAINING THEM AND THEIR USE AS PHARMACEUTICALS ELI LILLY AND COMPANY (US) 1982-09-22 EP disclosed
EP-0004173-A1 2,3-Dihydroimidazo (1,2-c) pyrimidines, their preparation, formulations containing them and their use as pharmaceuticals ELI LILLY AND COMPANY (US) 1979-09-19 EP disclosed