SCHEMBL11277817

SCHEMBL11277817

COC(=O)c1c(N)c(C)cn1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.41
GAA P10253 1/20 0.41
ALDH1A1 P00352 6/20 0.38
HSD17B10 Q99714 5/20 0.38
KDM4E B2RXH2 6/20 0.37
HPGD P15428 3/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MAPK1 P28482 1/20 0.37
NR4A2 P43354 1/20 0.37
DAPK3 O43293 1/20 0.36
JAK2 O60674 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
ABL1 P00519 1/20 0.36
CSF1R P07333 1/20 0.36
RET P07949 1/20 0.36
MET P08581 1/20 0.36
PDGFRA P16234 1/20 0.36
PRKACA P17612 1/20 0.36
LTK P29376 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11279081 0.82 LMNA (0.47) TSHRGAAALDH1A1HSD17B10KDM4E
SCHEMBL3938677 0.76 KDM4E (0.45) GAAALDH1A1HSD17B10KDM4EHPGD
SCHEMBL19503205 0.74 TDP1 (0.51) TSHRGAAALDH1A1KDM4EHPGD
SCHEMBL10970052 0.71 KDM4E (0.31) HSD17B10KDM4EHPGD
SCHEMBL22729485 0.69 BRD4 (0.39) TSHRGAAALDH1A1HSD17B10KDM4E
SCHEMBL14451934 0.69 ATM (0.38) TSHRGAAALDH1A1HSD17B10KDM4E
SCHEMBL11286998 0.69 KDM4E (0.46) TSHRGAAALDH1A1HSD17B10KDM4E
SCHEMBL29173842 0.67 KDM4E (0.37) TSHRGAAALDH1A1HSD17B10KDM4E
SCHEMBL11272207 0.67 KDM4E (0.45) TSHRGAAALDH1A1HSD17B10KDM4E
SCHEMBL10927533 0.66 BAZ2B (0.50) GAAALDH1A1HSD17B10KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4363816-A TREATMENT OF GASTROINTESTINAL DISORDERS BYK GULDEN LOMBERG CHEMISCHE FABRIK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1982-12-14 US disclosed