SCHEMBL11279359

SCHEMBL11279359

CN(C)C(=N)NC(=N)Nc1ccc(OCc2ccccc2)c(OCc2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 10/20 0.56
CYP19A1 P11511 6/20 0.49
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
ALOX12 P18054 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CTSV O60911 1/20 0.44
CTSL P07711 1/20 0.44
F2 P00734 1/20 0.43
F10 P00742 1/20 0.43
PRSS1 P07477 1/20 0.43
F7 P08709 1/20 0.43
MRGPRX1 Q96LB2 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11284130 0.88 CYP19A1 (0.44) C5AR1CYP19A1LMNA
SCHEMBL11283867 0.85 C5AR1 (0.58) C5AR1CYP19A1ALDH1A1LMNAMAPT
SCHEMBL11265836 0.84 C5AR1 (0.63) C5AR1ALDH1A1LMNAMAPTALOX12
SCHEMBL11596780 0.83 C5AR1 (0.62) C5AR1CYP19A1ALDH1A1LMNAMAPT
Hydrochloric Acid SCHEMBL11595019 0.82 C5AR1 (0.61) C5AR1CYP19A1ALDH1A1LMNAMAPT
SCHEMBL11253653 0.82 C5AR1 (0.55) C5AR1CYP19A1MAPTCTSVCTSL
SCHEMBL11264325 0.81 C5AR1 (0.60) C5AR1CYP19A1CTSVCTSLF2
SCHEMBL11274142 0.81 C5AR1 (0.62) C5AR1CYP19A1ALDH1A1LMNAMAPT
Hydrochloric Acid SCHEMBL11258213 0.81 C5AR1 (0.59) C5AR1CYP19A1CTSVCTSLF2
SCHEMBL11284600 0.80 C5AR1 (0.62) C5AR1CYP19A1ALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed