SCHEMBL11280893

SCHEMBL11280893

Cc1ccccc1NC(=N)N(C)C(=N)N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
SIGMAR1 Q99720 6/20 0.46
GRIN2D O15399 5/20 0.46
GRIN3B O60391 5/20 0.46
GRIN1 Q05586 5/20 0.46
GRIN2A Q12879 5/20 0.46
GRIN2B Q13224 5/20 0.46
GRIN2C Q14957 5/20 0.46
GRIN3A Q8TCU5 5/20 0.46
MEN1 O00255 1/20 0.46
PABPC1 P11940 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
KMT2A Q03164 1/20 0.46
EBP Q15125 1/20 0.46
TMEM97 Q5BJF2 1/20 0.46
HPGD P15428 4/20 0.46
ALDH1A1 P00352 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11558803 0.83 NPC1 (0.53) POLBNPC1RAB9ASIGMAR1GRIN2D
SCHEMBL11277630 0.81 GRIN2D (0.46) POLBSIGMAR1GRIN2DGRIN3BGRIN1
SCHEMBL467514 0.77 NPC1 (0.57) POLBNPC1RAB9ASIGMAR1GRIN2D
SCHEMBL29401646 0.77 NPC1 (0.57) POLBNPC1RAB9ASIGMAR1GRIN2D
SCHEMBL14868449 0.77 CA1 (0.39) ALOX15HPGDALDH1A1MAPTMAPK1
SCHEMBL14868313 0.77 TAS2R38 (0.45) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
Hydrochloric Acid SCHEMBL11234820 0.76 NPC1 (0.55) POLBNPC1RAB9ASIGMAR1GRIN2D
Guanidine SCHEMBL28181449 0.76 NPC1 (0.55) POLBNPC1RAB9ASIGMAR1GRIN2D
Hydrochloric Acid SCHEMBL31307094 0.76 NPC1 (0.55) POLBNPC1RAB9ASIGMAR1GRIN2D
SCHEMBL11279034 0.74 GAA (0.51) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4147804-A ANTIARRHYTHMIA AGENTS WILLIAM H. RORER, INC. (US) 1979-04-03 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed