SCHEMBL11282121

SCHEMBL11282121

CCCN1CC2(CCN(CCc3c[nH]c4ccccc34)CC2)OCC1=O

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.51
TACR2 P21452 1/20 0.49
TACR1 P25103 1/20 0.49
SIGMAR1 Q99720 1/20 0.49
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
DRD3 P35462 2/20 0.47
DRD2 P14416 1/20 0.47
DRD1 P21728 1/20 0.47
DRD4 P21917 1/20 0.47
DRD5 P21918 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11291802 0.99 HTR2A (0.50) HTR2ATACR2TACR1SIGMAR1RAB9A
SCHEMBL11281625 0.93 HTR2A (0.52) HTR2ATACR2TACR1SIGMAR1RAB9A
Hydrochloric Acid SCHEMBL11291237 0.92 HTR2A (0.51) HTR2ATACR2TACR1SIGMAR1RAB9A
SCHEMBL11286318 0.89 HTR2A (0.49) HTR2ATACR2TACR1SIGMAR1RAB9A
SCHEMBL11282509 0.88 SIGMAR1 (0.64) HTR2ATACR2TACR1SIGMAR1RAB9A
SCHEMBL18719630 0.88 TACR2 (0.62) HTR2ATACR2TACR1SIGMAR1
Hydrochloric Acid SCHEMBL11280625 0.87 SIGMAR1 (0.63) HTR2ATACR2TACR1SIGMAR1RAB9A
SCHEMBL11362813 0.86 TACR2 (0.62) TACR2TACR1
SCHEMBL18719628 0.83 SIGMAR1 (0.67) HTR2ATACR2TACR1SIGMAR1DRD3
SCHEMBL11368445 0.81 TACR2 (0.63) TACR2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0061333-A1 9-(2-(3-Indolyl)ethyl)-1-oxa-4,9-diazaspiro(5.5)undecan-3-ones SYNTEX (U.S.A.) INC. (US) 1982-09-29 EP claimed
US-4332804-A TREATMENT OF HYPERTENSION, CONGESTIVE HEART FAILURE, ARRHYTHMIA, MIGRAINE, VASOSPASTIC DISORDERS AND ASTHMA SYNTEX (U.S.A.) INC. (US) 1982-06-01 US claimed