SCHEMBL11282938

SCHEMBL11282938

O=C1NC2=Nc3cccc(Cl)c3CN2C1c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 7/20 0.68
PDE3A Q14432 7/20 0.68
LMNA P02545 1/20 0.68
CYP1A2 P05177 1/20 0.68
CYP3A4 P08684 1/20 0.68
CYP2D6 P10635 1/20 0.68
TSHR P16473 1/20 0.68
BLM P54132 1/20 0.68
CTSD P07339 1/20 0.44
KMT2A Q03164 2/20 0.36
ACHE P22303 1/20 0.36
MEN1 O00255 1/20 0.36
PDE2A O00408 1/20 0.36
P2RY12 Q9H244 1/20 0.36
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34
NR3C1 P04150 1/20 0.33
SLC6A3 Q01959 1/20 0.33
ALDH1A1 P00352 1/20 0.32
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11275717 0.99 PDE3B (0.67) PDE3BPDE3ALMNACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11287641 0.84 PDE3B (0.51) PDE3BPDE3ALMNACYP1A2CYP3A4
Quazinone SCHEMBL120976 0.81 PDE3B (1.00) PDE3BPDE3ALMNACYP1A2CYP3A4
Quazinone SCHEMBL2463520 0.81 PDE3B (1.00) PDE3BPDE3ALMNACYP1A2CYP3A4
SCHEMBL11283498 0.81 PDE3B (0.65) PDE3BPDE3ALMNACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11284634 0.80 PDE3B (0.64) PDE3BPDE3ALMNACYP1A2CYP3A4
Quazinone SCHEMBL11279841 0.80 PDE3B (0.97) PDE3BPDE3ALMNACYP1A2CYP3A4
SCHEMBL11278398 0.79 PDE3B (0.70) PDE3BPDE3ALMNACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11388525 0.78 PDE3B (0.68) PDE3BPDE3ALMNACYP1A2CYP3A4
SCHEMBL11279375 0.76 PDE3B (0.69) PDE3BPDE3ALMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0000718-B1 QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION, PHARMACEUTICAL PREPARATIONS AND THEIR PREPARATION F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1982-03-24 EP disclosed