SCHEMBL11286115

SCHEMBL11286115

COc1ccc2[nH]cc(CCN3CCC4(CC3)CNC(=O)CO4)c2c1

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.61
HTR1A P08908 8/20 0.56
ADRA2A P08913 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
ADRA1D P25100 1/20 0.49
ADRA1A P35348 1/20 0.49
ADRA1B P35368 1/20 0.49
DRD2 P14416 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11295861 0.84 HTR1D (0.50) HTR1A
SCHEMBL11021273 0.83 HTR2A (0.56) HTR2AHTR1AADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL11280259 0.82 HTR2A (0.55) HTR2AHTR1AADRA2AADRA2BADRA2C
SCHEMBL11281420 0.82 HTR2A (0.43) HTR2A
SCHEMBL11367195 0.80 HTR2A (0.53) HTR2AHTR1AADRA2ADRD2
SCHEMBL11288305 0.80 SIGMAR1 (0.53) ADRA2ADRD2
Hydrochloric Acid SCHEMBL11367589 0.79 HTR2A (0.53) HTR2AHTR1AADRA2ADRD2
SCHEMBL24723815 0.77 HTR2A (0.97) HTR2AHTR1AADRA2AADRA2BADRA2C
SCHEMBL25249411 0.77 HTR2A (1.00) HTR2AHTR1AADRA2AADRA2BADRA2C
SCHEMBL29633130 0.77 HTR2A (0.97) HTR2AHTR1AADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0061333-A1 9-(2-(3-Indolyl)ethyl)-1-oxa-4,9-diazaspiro(5.5)undecan-3-ones SYNTEX (U.S.A.) INC. (US) 1982-09-29 EP disclosed
US-4332804-A TREATMENT OF HYPERTENSION, CONGESTIVE HEART FAILURE, ARRHYTHMIA, MIGRAINE, VASOSPASTIC DISORDERS AND ASTHMA SYNTEX (U.S.A.) INC. (US) 1982-06-01 US disclosed