SCHEMBL11286306

SCHEMBL11286306

CCS(=O)(=O)c1ccc(C2CN=CN(C)C2)cc1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 8/20 0.39
RORC P51449 2/20 0.38
GAA P10253 2/20 0.37
PSIP1 O75475 2/20 0.36
CCL2 P13500 1/20 0.33
CNR2 P34972 3/20 0.33
APOBEC3A P31941 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11286859 0.79 NPC1 (0.33) RORCGAA
SCHEMBL11286241 0.77 SLC6A2 (0.34) TSHR
SCHEMBL11287270 0.75 SLC6A4 (0.34)
SCHEMBL11275552 0.75 NQO1 (0.41) RORCTSHR
SCHEMBL11287930 0.75 MAOB (0.35) GAA
SCHEMBL11277816 0.75 SRD5A1 (0.44)
SCHEMBL11282764 0.75 BRD4 (0.46) BRD4TSHR
SCHEMBL11083192 0.75 BRD4 (0.48) BRD4RORCGAAPSIP1
SCHEMBL11287661 0.74
Hydrochloric Acid SCHEMBL10674686 0.73 BRD4 (0.42) BRD4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed