SCHEMBL11290233

SCHEMBL11290233

COc1cc2c(cc1OC)CC(N(CCCCCC(=O)O)C(C)=O)CC2

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.40
NQO2 P16083 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
DRD2 P14416 2/20 0.38
DRD3 P35462 2/20 0.38
POLB P06746 1/20 0.37
MDM2 Q00987 2/20 0.36
MDM4 O15151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11323761 0.71 DRD2 (0.56) MTNR1AMTNR1BDRD2DRD3
SCHEMBL7800047 0.70 DRD2 (0.61) DRD2DRD3
SCHEMBL7800045 0.70 DRD2 (0.61) DRD2DRD3
SCHEMBL7333795 0.68 DRD3 (0.46) DRD2DRD3
SCHEMBL7333787 0.68 DRD3 (0.46) DRD2DRD3
SCHEMBL14882852 0.68 DRD2 (0.70) MTNR1AMTNR1BDRD2DRD3
SCHEMBL7342658 0.67 DRD2 (0.47) DRD2DRD3
SCHEMBL7342652 0.67 DRD2 (0.47) DRD2DRD3
Hydrochloric Acid SCHEMBL7330498 0.66 DRD3 (0.53) DRD2DRD3
SCHEMBL8768606 0.65 POLB (0.50) MAPK1MTNR1AMTNR1BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4256741-A INSECTICIDES, MITICIDES, APHIDICIDES VELSICOL CHEMICAL CORPORATION (US) 1981-03-17 US claimed
EP-0006217-B1 SUBSTITUTED AMINO ACIDS, THEIR USE AND PREPARATION, AND COMPOSITIONS CONTAINING THEM Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1982-03-31 EP disclosed
US-4243678-A GASTROINTESTINAL DISORDERS, LIVER DISORDERS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1981-01-06 US disclosed
EP-0006217-A1 Substituted amino acids, their use and preparation, and compositions containing them Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1980-01-09 EP disclosed