SCHEMBL11290589

SCHEMBL11290589

N#Cc1cc(O)cc(Nc2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.53
CYP3A4 P08684 1/20 0.53
ABCB1 P08183 3/20 0.47
ABCG2 Q9UNQ0 3/20 0.47
ABCC1 P33527 2/20 0.47
ALDH1A1 P00352 4/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
CXCR2 P25025 3/20 0.46
HSD17B10 Q99714 2/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
AR P10275 1/20 0.42
TAS2R14 Q9NYV8 1/20 0.42
ALOX15 P16050 1/20 0.41
ALOX12 P18054 1/20 0.41
PTGS1 P23219 1/20 0.41
SLC6A2 P23975 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28130804 0.87 ALDH1A1 (0.53) TSHRCYP3A4ABCB1ABCG2ALDH1A1
SCHEMBL10404276 0.80 CYP3A4 (0.71) TSHRCYP3A4ALDH1A1MAPTKDM4E
SCHEMBL25377834 0.79 ALDH1A1 (0.46) TSHRABCB1ABCG2ALDH1A1MAPT
SCHEMBL3750402 0.79 ALDH1A1 (0.46) TSHRABCB1ABCG2ALDH1A1MAPT
SCHEMBL12138925 0.78 ALDH1A1 (0.57) TSHRCYP3A4ABCB1ABCG2ALDH1A1
SCHEMBL6156438 0.77 ALDH1A1 (0.61) TSHRCYP3A4ABCG2ALDH1A1MAPT
Phenol SCHEMBL28795047 0.77 CA12 (0.52) TSHRCYP3A4ABCB1ABCG2ABCC1
SCHEMBL15145204 0.75 ALDH1A1 (0.53) TSHRCYP3A4ABCB1ABCG2ABCC1
SCHEMBL510240 0.74 ALDH1A1 (0.62) TSHRCYP3A4ABCB1ABCG2ABCC1
SCHEMBL9481712 0.74 ALDH1A1 (0.62) TSHRCYP3A4ABCB1ABCG2ABCC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0011254-B1 PROCESS FOR THE PREPARATION OF HYDRO-DIPHENYL AMINES BAYER AG (DE) 1982-01-13 EP disclosed
US-4265833-A CATALYTIC AMINATION OF A DIHYDROXYBENZENE WITH A PRIMARY AROMATIC AMINE BAYER AKTIENGESELLSCHAFT (DE) 1981-05-05 US disclosed
EP-0011254-A1 Process for the preparation of hydro-diphenyl amines BAYER AG (DE) 1980-05-28 EP disclosed