SCHEMBL11297155

SCHEMBL11297155

Nc1ccc(N2CCN(C(=O)O)CC2)cc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 1/20 0.49
RHEB Q15382 1/20 0.44
CASP6 P55212 1/20 0.44
GFER P55789 1/20 0.44
HTT P42858 3/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
MAPK1 P28482 3/20 0.42
LMNA P02545 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
KDM4E B2RXH2 2/20 0.42
GAA P10253 2/20 0.42
TSHR P16473 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MMP2 P08253 1/20 0.41
ADAMTS5 Q9UNA0 1/20 0.41
HTR1A P08908 1/20 0.41
HTR2A P28223 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17002237 0.86 GFER (0.62) CASP6GFERSMN1; SMN2KDM4EGAA
SCHEMBL3986081 0.85 IP6K1 (0.53) IP6K1CASP6GFERHTTMAPK1
SCHEMBL17265646 0.85 MAPT (0.52) IP6K1RHEBGFERHTTCA12
SCHEMBL23123759 0.83 IP6K1 (0.50) IP6K1CASP6GFERHTTMAPK1
SCHEMBL28094905 0.81 LMNA (0.43) HTTCA12CA1CA2CA9
SCHEMBL11299225 0.81 GAA (0.59) IP6K1CASP6GFERHTTMAPK1
SCHEMBL11299182 0.81 MAPT (0.51) IP6K1CASP6GFERHTTCA12
SCHEMBL11299382 0.81 IP6K1 (0.49) IP6K1CASP6GFERHTTMAPK1
SCHEMBL23293835 0.80 IP6K1 (0.59) IP6K1CASP6GFERHTTMAPK1
SCHEMBL18155100 0.80 IP6K1 (0.55) IP6K1CASP6GFERHTTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2665724-A1 BICYCLIC INHIBITORS OF ALK AbbVie Inc. (US) 2013-11-27 EP disclosed
WO-2012097682-A1 BICYCLIC INHIBITORS OF ALK ABBOTT LABORATORIES (US) 2012-07-26 WO disclosed