SCHEMBL1130795

SCHEMBL1130795

CC1(C)C(=O)N(c2ccc(OC(F)(F)F)c(NC(=O)CCN3CCOCC3)c2)C(=O)N1Cc1ccncc1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 5/20 0.45
WNT3A P56704 11/20 0.43
KMT2A Q03164 1/20 0.43
MAPK1 P28482 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KDR P35968 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL1130147 0.97 WNT3A (0.43) IGF1RWNT3AKMT2AMAPK1L3MBTL1
SCHEMBL1131486 0.93 IGF1R (0.47) IGF1RWNT3A
SCHEMBL1131471 0.93 IGF1R (0.47) IGF1RWNT3A
SCHEMBL1130966 0.93 IGF1R (0.46) IGF1R
SCHEMBL1129932 0.93 WNT3A (0.47) IGF1RWNT3A
SCHEMBL1131102 0.92 IGF1R (0.43) IGF1RWNT3AKDR
SCHEMBL1130336 0.92 IGF1R (0.46) IGF1RWNT3AKDR
SCHEMBL1129937 0.91 WNT3A (0.49) IGF1RWNT3A
SCHEMBL1131104 0.91 IGF1R (0.43) IGF1RWNT3AKDR
Trifluoroacetic Acid SCHEMBL1130075 0.91 IGF1R (0.44) IGF1RWNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773808-B1 NOVEL CYCLIC UREA DERIVATIVES, PREPARATION THEREOF AND PHARMACEUTICAL USE THEREOF AS KINASE INHIBITORS AVENTIS PHARMA SA (FR) 2011-02-16 EP claimed
US-7759379-B2 Cyclic urea derivatives, preparation thereof and pharmaceutical use thereof as kinase inhibitors AVENTIS PHARMA S.A. (FR) 2010-07-20 US claimed
US-20080004300-A1 Cyclic Urea Derivatives, Preparation Thereof And Pharmaceutical Use Thereof As Kinase Inhibitors AVENTIS PHARMA S.A. (FR) 2008-01-03 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080004300-A1 Cyclic Urea Derivatives, Preparation Thereof And Pharmaceutical Use Thereof As Kinase Inhibitors CDK2, CDK1, PRKAR2B IGF1R 446/4885WNT3A 3260/4885KMT2A 2500/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.