SCHEMBL1132765

SCHEMBL1132765

CO/C=C(/C(=O)O)c1ccccc1COc1cccc(C(F)(F)F)n1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 2/20 0.37
HCRTR2 O43614 4/20 0.35
HCRTR1 O43613 3/20 0.35
MRGPRX4 Q96LA9 2/20 0.35
HIF1A Q16665 1/20 0.34
SYK P43405 1/20 0.34
P2RX7 Q99572 1/20 0.33
OPRL1 P41146 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1132769 1.00 TAS2R14 (0.37) TAS2R14HCRTR2HCRTR1MRGPRX4HIF1A
SCHEMBL30748265 1.00 TAS2R14 (0.37) TAS2R14HCRTR2HCRTR1MRGPRX4HIF1A
Picoxystrobin SCHEMBL18977 0.91 HIF1A (0.39) TAS2R14HCRTR2HCRTR1MRGPRX4HIF1A
Picoxystrobin SCHEMBL675260 0.91 HIF1A (0.39) TAS2R14HCRTR2HCRTR1MRGPRX4HIF1A
Picoxystrobin SCHEMBL29377786 0.91 HIF1A (0.39) TAS2R14HCRTR2HCRTR1MRGPRX4HIF1A
SCHEMBL4648199 0.90 TAS2R14 (0.39) TAS2R14HCRTR2HCRTR1MRGPRX4HIF1A
Picoxystrobin SCHEMBL17701174 0.90 HIF1A (0.39) TAS2R14HCRTR2HCRTR1MRGPRX4HIF1A
SCHEMBL2259595 0.90 HCRTR2 (0.36) TAS2R14HCRTR2HCRTR1MRGPRX4P2RX7
SCHEMBL31287388 0.88 TAS2R14 (0.39) TAS2R14HCRTR2HCRTR1MRGPRX4P2RX7
SCHEMBL8726616 0.88 TAS2R14 (0.39) TAS2R14HCRTR2HCRTR1MRGPRX4P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 164 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180263243-A1 NOVEL PLANT PROTECTING COMPOSITIONS AND USES THEREOF FLECHSIG PATENT COMPANY LLC (CH) 2018-09-20 US claimed
EP-1450606-B1 SYNERGISTIC SEED TREATMENT COMPOSITIONS SYNGENTA PARTICIPATIONS AG (CH) 2011-02-16 EP claimed
EP-1267617-B2 FUNGICIDAL METHOD HERCULES INC (US) 2008-08-20 EP claimed
US-20060159772-A1 Fungicidal compositions ISAGRO S.P.A. (IT) 2006-07-20 US claimed
EP-1448057-B1 SEED TREATMENT COMPOSITIONS SYNGENTA PARTICIPATIONS AG (CH) 2006-05-24 EP claimed
WO-2006009967-A2 NOVEL ESTER AS USEFUL BROAD SPECTRUM FUNGICIDAL COMPOUNDS CORET JOEL MARCEL (US) 2006-01-26 WO claimed
US-20050282841-A1 Novel esters as useful broad spectrum fungicidal compounds CORET JOEL M 2005-12-22 US claimed
EP-1565057-A2 FUNGICIDAL COMPOSITIONS CONTAINING AT LEAST ONE SALT OF PHOSPHOROUS ACID AND AT LEAST A SECOND FUNGICIDAL COMPONENT ISAGRO S.p.A. (IT) 2005-08-24 EP claimed
US-20050065031-A1 Synergistic seed treatment compositions LANXESS CORPORATION 2005-03-24 US claimed
US-20050043176-A1 Seed treatment compositions SYNGENTA CROP PROTECTION, INC. 2005-02-24 US claimed
US-6653258-B1 Pyridinyl-substituted- methyl 3-methoxy-2-phenylacrylate derivatives; agricultural miticides and nematocides SYNGENTA LIMITED (GB) 2003-11-25 US claimed
WO-2003045150-A2 SEED TREATMENT COMPOSITIONS SYNGENTA PARTICIPATIONS AG (CH) 2003-06-05 WO claimed
WO-2003045146-A1 SEED TREATMENT COMPOSITIONS SYNGENTA PARTICIPATIONS AG (CH) 2003-06-05 WO claimed
WO-2003045147-A1 SYNERGISTIC SEED TREATMENT COMPOSITIONS SYNGENTA PARTICIPATIONS AG (CH) 2003-06-05 WO claimed
EP-1267617-A2 FUNGICIDAL METHOD HERCULES INCORPORATED (US) 2003-01-02 EP claimed
US-20020108730-A1 FUNGICIDAL METHOD SOLENIS TECHNOLOGIES, L.P. 2002-08-15 US claimed
US-6428654-B1 COMBINING FUNGICIDE COMPRISING STROBILURIN WITH AQUEOUS SYSTEM COMPRISING PAPERMAKING STOCK TANK, PULP REFINER, STOCK CHEST, FLOW BOX, FURNISH OR WET-LAP TO CONTROL GROWTH OF FUNGI OR MILDEW HERCULES INCORPORATED 2002-08-06 US claimed
US-6338742-B1 LOW MELTING AGROCHEMICALS AS SUSPENSION CONCENTRATES, EUTECTIC MIXTURE OF FUNGICIDES METHYL-2-(2-(6-(TRIFLUOROMETHYL) PYRIDIN-2-YLOXYMETHYL) PHENYL)-3-METHOXYACRYLATE AND AZOXYSTROBIN, SUBJECTING EMULSION TO ULTRASONIC VIBRATION. SYNGENTA LIMITED (GB) 2002-01-15 US claimed
WO-2001077026-A2 FUNGICIDAL METHOD HERCULES INCORPORATED (US) 2001-10-18 WO claimed
EP-0946232-B1 CRYSTALLISATION PROCESS SYNGENTA LTD (GB) 2001-08-22 EP claimed