SCHEMBL11342016

SCHEMBL11342016

Fc1ccc(CN2CCNCC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.66
CXCR4 P61073 11/20 0.65
MEN1 O00255 1/20 0.65
CHRM2 P08172 1/20 0.65
CHRM1 P11229 1/20 0.65
ADRA2C P18825 1/20 0.65
CCR2 P41597 1/20 0.65
CXCL12 P48061 1/20 0.65
BLM P54132 1/20 0.65
KMT2A Q03164 1/20 0.65
TDP1 Q9NUW8 1/20 0.65
HRH3 Q9Y5N1 1/20 0.65
ALDH1A1 P00352 1/20 0.53
POLB P06746 1/20 0.53
MAPT P10636 1/20 0.53
SLC6A2 P23975 1/20 0.53
SLC6A4 P31645 1/20 0.53
SLC6A3 Q01959 1/20 0.53
KCNH2 Q12809 1/20 0.53
HTR6 P50406 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL211040 1.00 SIGMAR1 (0.66) SIGMAR1CXCR4MEN1CHRM2CHRM1
Hydrochloric Acid SCHEMBL3062972 0.98 CXCR4 (0.66) SIGMAR1CXCR4MEN1CHRM2CHRM1
Hydrochloric Acid SCHEMBL6291076 0.98 CXCR4 (0.66) SIGMAR1CXCR4MEN1CHRM2CHRM1
SCHEMBL2003768 0.93 CXCR4 (0.77) SIGMAR1CXCR4MEN1CHRM2CHRM1
Hydrochloric Acid SCHEMBL209072 0.91 CXCR4 (0.78) SIGMAR1CXCR4MEN1CHRM2CHRM1
SCHEMBL2233118 0.90 SIGMAR1 (0.54) SIGMAR1CXCR4MEN1CHRM2CHRM1
SCHEMBL1259387 0.87 CXCR4 (0.81) SIGMAR1CXCR4MEN1CHRM2CHRM1
Hydrochloric Acid SCHEMBL5573232 0.87 CXCR4 (0.78) SIGMAR1CXCR4MEN1CHRM2CHRM1
SCHEMBL2233922 0.86 HRH3 (0.64) SIGMAR1CXCR4MEN1CHRM2CHRM1
Bromide SCHEMBL1257550 0.85 CXCR4 (0.78) SIGMAR1CXCR4MEN1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4243805-A 3 Fluoro-10-piperazino-8-substituted 10,11-dihydrodibenzo-(bf) thiepins and method for the preparation thereof SPOFA, SPOJENE PODNIKY PRO ZDRAVOTNICKOU VYROBU (CS) 1981-01-06 US disclosed