SCHEMBL11348371

SCHEMBL11348371

Cc1ccc2c(c1)C(=O)c1nn[nH]c1C2=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.50
MAOB P27338 1/20 0.50
ELANE P08246 1/20 0.49
USP8 P40818 1/20 0.44
USP7 Q93009 1/20 0.44
RAB9A P51151 2/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
LCK P06239 1/20 0.39
NQO1 P15559 2/20 0.36
POR P16435 2/20 0.36
CA9 Q16790 2/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA7 P43166 1/20 0.35
ROS1 P08922 1/20 0.35
CDK5 Q00535 1/20 0.35
ACVR1 Q04771 1/20 0.35
LRRK2 Q5S007 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11346081 0.83 NQO1 (0.33) MAOBRAB9AMAPTSMN1; SMN2NQO1
SCHEMBL11345791 0.81 NQO1 (0.33) NQO1POR
SCHEMBL11345788 0.81 NQO1 (0.33) NQO1POR
SCHEMBL11353687 0.81 USP8 (0.44) MAOBUSP8USP7RAB9AMAPT
SCHEMBL11352822 0.80 USP8 (0.48) MAOAMAOBUSP8RAB9AMAPT
SCHEMBL11020695 0.79 POLB (0.52) MAOAUSP8USP7RAB9AMAPT
SCHEMBL24976667 0.75 ELANE (0.42) MAOBELANEUSP8USP7RAB9A
SCHEMBL24976533 0.75 ELANE (0.42) MAOBELANEUSP8USP7RAB9A
SCHEMBL11359550 0.73 TDP2 (0.50) ELANEUSP8USP7RAB9ASMN1; SMN2
SCHEMBL583153 0.72 ELANE (0.86) MAOAMAOBELANEUSP8USP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0002310-A1 4,9-Dihydro-4,9-dioxo-1H-naphtho(2,3-d) triazoles, their preparation and antiallergic compositions containing them BEECHAM GROUP PLC (GB) 1979-06-13 EP claimed
EP-0002310-B1 4,9-DIHYDRO-4,9-DIOXO-1H-NAPHTHO(2,3-D) TRIAZOLES, THEIR PREPARATION AND ANTIALLERGIC COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1981-06-24 EP disclosed
US-4263309-A ASTHMA, HAY FEVER, RHINITIS BEECHAM GROUP LIMITED (GB) 1981-04-21 US disclosed
EP-0002310-A1 4,9-Dihydro-4,9-dioxo-1H-naphtho(2,3-d) triazoles, their preparation and antiallergic compositions containing them BEECHAM GROUP PLC (GB) 1979-06-13 EP disclosed