SCHEMBL1137261

SCHEMBL1137261

Cc1ccn(Cc2ccccc2)c(=O)c1C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.56
SMN1; SMN2 Q16637 2/20 0.51
TP53 P04637 2/20 0.51
HTT P42858 2/20 0.51
KDM4E B2RXH2 1/20 0.51
CYP2D6 P10635 1/20 0.51
POLB P06746 3/20 0.50
BRD4 O60885 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
MAPK14 Q16539 2/20 0.50
BRD2 P25440 1/20 0.50
BRD3 Q15059 1/20 0.50
BRDT Q58F21 1/20 0.50
EGLN1 Q9GZT9 2/20 0.48
FAAH O00519 1/20 0.47
CNR1 P21554 1/20 0.47
CNR2 P34972 1/20 0.47
MAPT P10636 2/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25612867 0.87 CNR2 (0.62) NOTUMSMN1; SMN2TP53KDM4EMEN1
SCHEMBL11608258 0.83 KDM4E (0.47) SMN1; SMN2TP53HTTKDM4EPOLB
SCHEMBL28069907 0.83 NOTUM (0.62) NOTUMSMN1; SMN2TP53HTTKDM4E
SCHEMBL12502932 0.79 NOTUM (0.55) NOTUMKDM4EBRD4MAPK14BRD2
SCHEMBL4685054 0.78 MAPK14 (0.52) NOTUMSMN1; SMN2TP53HTTKDM4E
SCHEMBL6652306 0.78 MAPK14 (0.60) NOTUMSMN1; SMN2TP53HTTKDM4E
SCHEMBL12502722 0.76 NOTUM (0.58) NOTUMSMN1; SMN2KDM4EPOLBBRD4
SCHEMBL29639001 0.76 NOTUM (0.42) NOTUMSMN1; SMN2TP53HTTKDM4E
SCHEMBL16509736 0.75 BRD4 (0.56) SMN1; SMN2TP53HTTKDM4ECYP2D6
SCHEMBL3175610 0.75 NOTUM (0.46) NOTUMSMN1; SMN2TP53HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737451-B1 MONOCYCLIC HETEROCYCLES AS KINASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2011-02-23 EP disclosed