SCHEMBL11375646

SCHEMBL11375646

CC(C)(C(=O)O)C1(O)CCN(Cc2ccccc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 2/20 0.59
POLB P06746 1/20 0.57
CCR3 P51677 1/20 0.57
CYP2D6 P10635 4/20 0.56
CHRM2 P08172 1/20 0.51
CHRM3 P20309 1/20 0.51
ALDH1A1 P00352 3/20 0.50
CYP3A4 P08684 2/20 0.50
HSD17B10 Q99714 1/20 0.50
DRD2 P14416 1/20 0.50
DRD4 P21917 1/20 0.50
DRD3 P35462 1/20 0.50
TSHR P16473 1/20 0.49
KMT2A Q03164 2/20 0.49
LMNA P02545 1/20 0.49
SIGMAR1 Q99720 1/20 0.49
USP2 O75604 1/20 0.48
MAPK1 P28482 1/20 0.48
MEN1 O00255 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17101429 0.85 CYP2D6 (0.51) OPRL1POLBCCR3CYP2D6CHRM2
SCHEMBL596787 0.84 CYP2D6 (0.55) OPRL1POLBCYP2D6CHRM2CHRM3
SCHEMBL16973869 0.83 OPRL1 (0.59) OPRL1POLBCCR3CYP2D6CHRM2
SCHEMBL4484154 0.78 OPRL1 (0.61) OPRL1POLBCCR3CYP2D6CHRM2
SCHEMBL11362333 0.77 MEN1 (0.54) ALDH1A1KMT2ASIGMAR1MEN1
SCHEMBL1147211 0.76 OPRL1 (0.63) OPRL1POLBCCR3CYP2D6CHRM2
SCHEMBL31334693 0.76 NPFFR1 (0.53) OPRL1POLBCCR3CYP2D6CHRM2
SCHEMBL653329 0.76 OPRL1 (0.67) OPRL1POLBCCR3CYP2D6CHRM2
SCHEMBL28548988 0.76 OPRL1 (0.71) OPRL1POLBCCR3CYP2D6CHRM2
Hydrochloric Acid SCHEMBL25235306 0.75 POLB (0.64) OPRL1POLBCCR3CYP2D6CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4255432-A ANTIHYPERTENSIVE AGENTS, ANTIHISTAMINES, BRONCHODILATOR AGENTS, ANTIVASOSPASTIC AGENTS SYNTEX (U.S.A.) INC. (US) 1981-03-10 US disclosed
US-4244961-A 1-Oxa-3,8-diazaspiro[4.5]decan-2-ones antihypertensive agents SYNTEX (U.S.A.) INC. (US) 1981-01-13 US disclosed