SCHEMBL11384331

SCHEMBL11384331

Fc1ccc(-c2ccc3nncn3c2)cc1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.64
SCN5A Q14524 2/20 0.62
TGFBR1 P36897 1/20 0.57
DNMT1 P26358 1/20 0.53
PIK3CA P42336 1/20 0.51
ALDH1A3 P47895 4/20 0.49
MLLT1 Q03111 2/20 0.45
ADORA2A P29274 2/20 0.41
ADORA2B P29275 2/20 0.41
ADORA1 P30542 2/20 0.41
EGLN1 Q9GZT9 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
MAPK1 P28482 1/20 0.39
MLLT3 P42568 1/20 0.38
DYRK1A Q13627 1/20 0.36
ALDH1A2 O94788 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15008043 0.84 MAPK14 (0.54) MAPK14SCN5ATGFBR1DNMT1PIK3CA
SCHEMBL11379662 0.83 SCN5A (0.59) MAPK14SCN5ATGFBR1DNMT1PIK3CA
SCHEMBL2538610 0.82 SCN5A (0.51) MAPK14SCN5ATGFBR1DNMT1PIK3CA
SCHEMBL11474506 0.81 SCN5A (0.58) MAPK14SCN5ATGFBR1DNMT1PIK3CA
SCHEMBL11476887 0.81 SCN5A (0.58) MAPK14SCN5ATGFBR1DNMT1PIK3CA
SCHEMBL11486274 0.81 SCN5A (0.58) MAPK14SCN5ATGFBR1DNMT1PIK3CA
SCHEMBL19806542 0.78 MAPK14 (0.56) MAPK14SCN5ATGFBR1DNMT1PIK3CA
SCHEMBL11475951 0.77 SCN5A (0.57) MAPK14SCN5ATGFBR1DNMT1NPC1
SCHEMBL11491065 0.77 SCN5A (0.66) MAPK14SCN5ADNMT1PIK3CAALDH1A3
SCHEMBL2538823 0.77 SCN5A (0.50) MAPK14SCN5ATGFBR1DNMT1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4244953-A Substituted 6-phenyl-5,6,7,8-tetrahydro-1,2,4-triazolo-[4,3-a]pyridines AMERICAN CYANAMID COMPANY (US) 1981-01-13 US disclosed
US-4209626-A Substituted 6-phenyl-1,2,4-triazolo[4,3-a]pyridines AMERICAN CYANAMID COMPANY (US) 1980-06-24 US disclosed