SCHEMBL11389554

SCHEMBL11389554

CCOC(=O)C1Cc2ccccc2N1CC

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1D1 P20393 4/20 0.49
ALDH1A1 P00352 1/20 0.44
NOTUM Q6P988 1/20 0.44
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 1/20 0.43
BCL2 P10415 1/20 0.42
BAD Q92934 1/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10907233 0.87 NR1D1 (0.48) NR1D1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL11392205 0.86 NOTUM (0.48) NR1D1ALDH1A1NOTUMKDM4E
SCHEMBL27900298 0.85 NR1D1 (0.45) NR1D1ALDH1A1NOTUMTP53CYP1A2
SCHEMBL8429535 0.84 PRKCD (0.48) NR1D1ALDH1A1
SCHEMBL23343522 0.84 NR1D1 (0.50) NR1D1NOTUMTP53
SCHEMBL4959583 0.84 NR1D1 (0.50) NR1D1NOTUMTP53
SCHEMBL11821195 0.83 NR1D1 (0.46) NR1D1ALDH1A1NOTUMTP53BCL2
SCHEMBL12643017 0.83 DRD4 (0.52) NR1D1
SCHEMBL17461323 0.83 NR1D1 (0.49) NR1D1ALDH1A1NOTUMTP53KDM4E
SCHEMBL13068180 0.83 NR1D1 (0.49) NR1D1NOTUMTP53BCL2BAD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9763955-B2 Methods and compositions for decreasing gastric emptying PURDUE PHARMA L.P. (US) 2017-09-19 US disclosed
WO-2017027710-A1 ELECTRON DONOR FOR POLYOLEFIN POLYMERIZATION CATALYSTS AND USES THEREOF W.R. GRACE & CO.-CONN. (US) 2017-02-16 WO disclosed
WO-2014151393-A2 CARBOXAMIDE DERIVATIVES AND USE THEREOF PURDUE PHARMA L.P. (US) 2014-09-25 WO disclosed
US-4260628-A 2-Guanidinomethyl-indolines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1981-04-07 US disclosed