SCHEMBL11396129

SCHEMBL11396129

NC(C(=O)O)c1ccc(O)c(F)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 7/20 0.64
KDM4E B2RXH2 7/20 0.64
TDP1 Q9NUW8 6/20 0.64
ALDH1A1 P00352 4/20 0.64
HPGD P15428 4/20 0.64
CYP2C9 P11712 4/20 0.64
GRM1 Q13255 3/20 0.64
MEN1 O00255 3/20 0.64
KMT2A Q03164 3/20 0.64
CYP2C19 P33261 3/20 0.64
GRM2 Q14416 2/20 0.59
CYP2D6 P10635 1/20 0.53
GRM8 O00222 1/20 0.53
GRM6 O15303 1/20 0.53
SLC6A2 P23975 1/20 0.53
SLC6A4 P31645 1/20 0.53
DRD3 P35462 1/20 0.53
GRM4 Q14833 1/20 0.53
LMNA P02545 3/20 0.46
BLM P54132 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11451469 0.85 HSD17B10 (0.46) HSD17B10KDM4ETDP1ALDH1A1HPGD
SCHEMBL11386312 0.85 HSD17B10 (0.46) HSD17B10KDM4ETDP1ALDH1A1HPGD
SCHEMBL31091372 0.85 HSD17B10 (0.56) HSD17B10KDM4ETDP1ALDH1A1HPGD
SCHEMBL11386310 0.84 HSD17B10 (0.45) HSD17B10KDM4ETDP1ALDH1A1HPGD
SCHEMBL3478437 0.82 TDP1 (0.70) HSD17B10KDM4ETDP1ALDH1A1HPGD
SCHEMBL10723439 0.82 TDP1 (0.70) HSD17B10KDM4ETDP1ALDH1A1HPGD
SCHEMBL449665 0.82 TDP1 (0.70) HSD17B10KDM4ETDP1ALDH1A1HPGD
Bromide SCHEMBL11670638 0.81 TDP1 (0.68) HSD17B10KDM4ETDP1ALDH1A1HPGD
SCHEMBL12498905 0.80 HSD17B10 (0.51) HSD17B10KDM4ETDP1ALDH1A1HPGD
SCHEMBL30468550 0.80 HSD17B10 (0.51) HSD17B10KDM4ETDP1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4257947-A INTERMEDIATES FOR ANTIBACTERIAL CEPHALOSPORINS SMITHKLINE CORPORATION (US) 1981-03-24 US disclosed
US-4236001-A 7β-Acyloxy-3-heterocyclicthiomethyl cephalosporins SMITHKLINE CORPORATION (US) 1980-11-25 US disclosed
US-4218564-A 7β-Hydroxy-3-heterocyclicthio-methyl cephalosporin intermediates SMITHKLINE CORPORATION (US) 1980-08-19 US disclosed
US-4166816-A CYCLIZATION SMITHKLINE CORPORATION (US) 1979-09-04 US disclosed
US-4158733-A 7β-Acyloxy-3-acetoxymethyl cephalosporins SMITHKLINE CORPORATION (US) 1979-06-19 US disclosed
US-4131734-A 7β-Acyloxy-3-heterocyclicthiomethyl cephalosporins SMITHKLINE CORPORATION (US) 1978-12-26 US disclosed
US-4103086-A 8-Oxo-4-thia-1-azabicyclo (4.2.0)-oct-2-ene derivatives SMITHKLINE CORPORATION (US) 1978-07-25 US disclosed
US-4072674-A FOR CEPHALOSPORIN CONGENERS SMITHKLINE CORPORATION (US) 1978-02-07 US disclosed
US-4020057-A 7β-Acyloxy cephalosporins SMITHKLINE CORPORATION (US) 1977-04-26 US disclosed