SCHEMBL11397192

SCHEMBL11397192

Cc1nnc(CBr)n1-c1ccccc1C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MYC P01106 7/20 0.54
NR4A1 P22736 1/20 0.54
POLB P06746 2/20 0.47
ALDH1A1 P00352 2/20 0.45
SETDB1 Q15047 1/20 0.42
TSHR P16473 1/20 0.41
ALOX15 P16050 1/20 0.40
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38
NOTUM Q6P988 1/20 0.38
APEX1 P27695 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11400787 0.86 MYC (0.50) MYCNR4A1POLBALDH1A1TSHR
SCHEMBL11402376 0.85 MYC (0.57) MYCPOLBALDH1A1SETDB1TSHR
SCHEMBL11404295 0.83 MYC (0.48) MYCNR4A1POLBALDH1A1ALOX15
SCHEMBL11404481 0.82 MYC (0.59) MYCNR4A1SETDB1APEX1
SCHEMBL11405951 0.82 MYC (0.47) MYCNR4A1POLBALDH1A1TSHR
SCHEMBL11400991 0.81 MYC (0.42) MYCNR4A1ALDH1A1SETDB1NOTUM
SCHEMBL11398198 0.81 MYC (0.58) MYCNR4A1ALDH1A1SETDB1TSHR
SCHEMBL11397291 0.81 MYC (0.49) MYCNR4A1POLBALDH1A1SETDB1
SCHEMBL11825290 0.77 MAPT (0.46) MYCNR4A1POLBALDH1A1SETDB1
SCHEMBL11826302 0.76 HTT (0.50) MYCNR4A1ALDH1A1SETDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4296239-A Amino-4H-s-triazolo[4,3-a][1,4]benzodiazepines THE UPJOHN COMPANY (US) 1981-10-20 US disclosed
US-4180668-A Piperidino-4H-s-triazolo[4,3-a][1,4]benzodiazepines THE UPJOHN COMPANY (US) 1979-12-25 US disclosed