SCHEMBL11433713

SCHEMBL11433713

OC(Cc1ncc[nH]1)c1ccc2ccccc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.49
ADRA2B P18089 2/20 0.49
ADRA2C P18825 2/20 0.49
CYP2D6 P10635 5/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
AOC3 Q16853 1/20 0.44
CYP1A2 P05177 1/20 0.44
TSHR P16473 1/20 0.44
HIF1A Q16665 1/20 0.44
UGT2B7 P16662 1/20 0.42
TAAR1 Q96RJ0 3/20 0.41
SLC6A2 P23975 5/20 0.40
SLC6A4 P31645 5/20 0.40
SLC6A3 Q01959 5/20 0.40
KCNH2 Q12809 4/20 0.40
CYP3A4 P08684 4/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6299755 0.82 TAAR1 (0.51) CYP2D6MEN1KMT2ATSHRTAAR1
SCHEMBL6299922 0.82 TAAR1 (0.51) CYP2D6MEN1KMT2ATSHRTAAR1
SCHEMBL11433350 0.80 AOC3 (0.49) ADRA2AADRA2BADRA2CCYP2D6AOC3
SCHEMBL11296792 0.78 TAAR1 (0.42) MEN1KMT2ATAAR1HTR1A
SCHEMBL11289983 0.77 TAAR1 (0.44) TAAR1HTR1A
SCHEMBL3528465 0.75 TAAR1 (0.39) MEN1KMT2ATAAR1
SCHEMBL3529536 0.75 TAAR1 (0.39) ADRA2AADRA2BADRA2CTAAR1
SCHEMBL3913688 0.75 TAAR1 (0.39) MEN1KMT2ATAAR1
SCHEMBL8488446 0.75 TAAR1 (0.37) ADRA2AADRA2BADRA2CCYP2D6CYP1A2
SCHEMBL11566236 0.74 ADRA2A (0.54) ADRA2AADRA2BADRA2CCYP2D6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0013786-A1 Imidazole derivatives, pharmaceutical compositions containing them and their preparation SYNTEX (U.S.A.) INC. (US) 1980-08-06 EP disclosed
EP-0001926-A1 1-(Naphthylethyl)imidazole derivatives, their preparation, and pharmaceutical compositions containing them SYNTEX (U.S.A.) INC. (US) 1979-05-16 EP disclosed