SCHEMBL11449643

SCHEMBL11449643

CN1CCCC1CCOc1ccccc1O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 3/20 0.55
CHRNA3 P32297 3/20 0.55
SLC22A1 O15245 1/20 0.49
MLNR O43193 1/20 0.49
NR1I2 O75469 1/20 0.49
TP53 P04637 1/20 0.49
ADRB2 P07550 1/20 0.49
CHRM2 P08172 1/20 0.49
CHRM4 P08173 1/20 0.49
ADRB1 P08588 1/20 0.49
CYP3A4 P08684 1/20 0.49
HTR1A P08908 1/20 0.49
CHRM5 P08912 1/20 0.49
ADRA2A P08913 1/20 0.49
CYP2D6 P10635 1/20 0.49
CHRM1 P11229 1/20 0.49
CYP2C9 P11712 1/20 0.49
DRD2 P14416 1/20 0.49
TSHR P16473 1/20 0.49
ADRA2B P18089 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11447617 0.97 CHRNB4 (0.52) CHRNB4CHRNA3SLC22A1MLNRNR1I2
Hydrochloric Acid SCHEMBL8703569 0.86 TP53 (0.49) CHRNB4CHRNA3SLC22A1MLNRNR1I2
SCHEMBL14578238 0.85 CHRNB4 (0.61) CHRNB4CHRNA3SLC22A1MLNRNR1I2
SCHEMBL11448305 0.84 TDP1 (0.57) CHRNB4CHRNA3CYP2D6CYP2C19CHRNB2
SCHEMBL11455709 0.84 CHRNB4 (0.76) CHRNB4CHRNA3HTR2ACHRNB2CHRNA4
SCHEMBL11466714 0.83 TSHR (0.55) CHRNB4CHRNA3SLC22A1MLNRNR1I2
SCHEMBL11447873 0.83 CHRNB4 (0.55) CHRNB4CHRNA3CYP3A4CYP2D6CYP2C9
SCHEMBL14578289 0.83 CHRNB4 (0.58) CHRNB4CHRNA3SLC22A1MLNRNR1I2
SCHEMBL11448129 0.83 CHRNB4 (0.55) CHRNB4CHRNA3CHRNB2CHRNA4LMNA
SCHEMBL11449219 0.82 TDP1 (0.58) CHRNB4CHRNA3ADRA2ACYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4225608-A ANTIDEPRESSANTS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1980-09-30 US disclosed
EP-0004288-A2 Phenoxyalkyl amines, pharmaceutical compositions containing them, and process for their preparation MERCK PATENT GmbH (DE) 1979-10-03 EP disclosed