SCHEMBL1145495

SCHEMBL1145495

Cc1ncc(C#N)c(Nc2ccc3[nH]ccc3c2)c1-c1cccs1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PRKCQ Q04759 18/20 0.55
PRKCD Q05655 9/20 0.55
LYN P07948 1/20 0.55
EGFR P00533 2/20 0.49
FLT1 P17948 2/20 0.49
PRKCH P24723 1/20 0.48
PRKCE Q02156 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1146158 0.83 PRKCQ (0.58) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL1145652 0.83 PRKCQ (0.64) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2975707 0.82 PRKCQ (0.60) PRKCQPRKCDLYNEGFRFLT1
SCHEMBL1146429 0.80 PRKCQ (0.61) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL1146156 0.80 PRKCQ (0.54) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL1146269 0.80 PRKCQ (0.54) PRKCQPRKCDLYNFLT1PRKCH
SCHEMBL1146471 0.79 PRKCQ (0.59) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL1146524 0.78 PRKCQ (0.54) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL1146331 0.78 PRKCQ (0.55) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL1146445 0.78 PRKCQ (0.71) PRKCQPRKCDLYNPRKCHPRKCE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110028455-A1 Indole-substituted 3-cyanopyridines As Kinase Inhibitors WYETH LLC (US) 2011-02-03 US claimed
EP-2229376-A1 INDOLE-SUBSTITUTED 3-CYANOPYRIDINES AS KINASE INHIBITORS Wyeth LLC (US) 2010-09-22 EP claimed
WO-2009076571-A1 INDOLE-SUBSTITUTED 3-CYANOPYRIDINES AS KINASE INHIBITORS WYETH (US) 2009-06-18 WO claimed
US-20110028455-A1 Indole-substituted 3-cyanopyridines As Kinase Inhibitors WYETH LLC (US) 2011-02-03 US disclosed
US-20110028455-A1 Indole-substituted 3-cyanopyridines As Kinase Inhibitors WYETH LLC (US) 2011-02-03 US disclosed
US-20110028455-A1 Indole-substituted 3-cyanopyridines As Kinase Inhibitors WYETH LLC (US) 2011-02-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110028455-A1 Indole-substituted 3-cyanopyridines As Kinase Inhibitors CNKSR1, CSNK1G3, GRK3 PRKCQ 324/4885PRKCD 291/4885LYN 133/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.