SCHEMBL11470945

SCHEMBL11470945

O=C(O)c1cccc(-c2ccnc3ccnn23)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 9/20 0.52
KDM5B Q9UGL1 8/20 0.52
KDM5A P29375 7/20 0.52
KDM4A O75164 1/20 0.52
KMO O15229 2/20 0.46
PDE4D Q08499 1/20 0.46
KEAP1 Q14145 1/20 0.46
NPC1 O15118 1/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
PIK3CD O00329 1/20 0.44
CD74 P04233 1/20 0.43
MIF P14174 1/20 0.43
DYRK3 O43781 1/20 0.43
DYRK1A Q13627 1/20 0.43
DYRK2 Q92630 1/20 0.43
DYRK1B Q9Y463 1/20 0.43
KDM2B Q8NHM5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11463687 0.78 EGLN2 (0.58) KDM4CKDM5BKDM5ANPC1LMNA
SCHEMBL10761987 0.78 KDM4E (0.41) KDM4CKDM5BKDM5AKDM4APDE4D
SCHEMBL30740531 0.77 KDM5A (0.52) KDM4CKDM5BKDM5AKDM4AKMO
SCHEMBL940183 0.77 KDM5A (0.52) KDM4CKDM5BKDM5AKDM4AKMO
SCHEMBL3155417 0.76 KDM4E (0.54) KDM4CKDM5BKDM5AKDM4APDE4D
SCHEMBL11473783 0.74 EGLN2 (0.68)
SCHEMBL5946455 0.74 DYRK3 (0.47) PDE4DDYRK3DYRK1ADYRK2DYRK1B
SCHEMBL5946454 0.73 EGLN2 (0.39) PDE4DNPC1LMNAMAPTRAB9A
SCHEMBL6071500 0.71 EGLN2 (0.51) PDE4DMAPTRAB9ADYRK1AFYN
SCHEMBL21310947 0.71 DYRK1A (0.50) KDM4CKDM5BKDM5AKDM4AKMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4236005-A ANTIANXIETY AMERICAN CYANAMID COMPANY (US) 1980-11-25 US disclosed
US-4178449-A Pyrazolo[1,5-a]pyrimidines and imidazo-[1,5-a]pyrimidines AMERICAN CYANAMID COMPANY (US) 1979-12-11 US disclosed