SCHEMBL6071500

SCHEMBL6071500

CCOc1cccc(-c2ccnc3ccnn23)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 1/20 0.51
FYN P06241 2/20 0.47
PDE4D Q08499 1/20 0.46
DYRK1A Q13627 1/20 0.46
BRD4 O60885 1/20 0.45
BRD2 P25440 1/20 0.45
CREBBP Q92793 1/20 0.45
S1PR1 P21453 3/20 0.44
AAK1 Q2M2I8 1/20 0.43
MAPT P10636 4/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
SIRT1 Q96EB6 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
NOTUM Q6P988 1/20 0.42
TDP1 Q9NUW8 2/20 0.42
KDM4E B2RXH2 2/20 0.41
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16331500 0.83 DYRK1A (0.67) EGLN2FYNDYRK1AS1PR1MAPT
SCHEMBL6071178 0.77 MAPKAPK2 (0.42) EGLN2FYNDYRK1AAAK1MAPT
SCHEMBL21575262 0.76 AAK1 (0.49) EGLN2CREBBPS1PR1AAK1MAPT
SCHEMBL6071200 0.76 DYRK1A (0.49) EGLN2FYNPDE4DDYRK1AAAK1
SCHEMBL11463687 0.74 EGLN2 (0.58) EGLN2FYNDYRK1AMAPTALDH1A1
SCHEMBL21575275 0.74 AAK1 (0.47) EGLN2AAK1SMN1; SMN2
SCHEMBL21575311 0.74 AAK1 (0.52) EGLN2S1PR1AAK1RXRARXRB
SCHEMBL11473783 0.73 EGLN2 (0.68) EGLN2KDM4E
SCHEMBL3155417 0.73 KDM4E (0.54) EGLN2FYNPDE4DAAK1MAPT
SCHEMBL10553161 0.72 KDM4E (0.57) EGLN2FYNPDE4DDYRK1AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060063784-A1 Method of using substituted pyrazolo [1,5-a] pyrimidines WYETH 2006-03-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060063784-A1 Method of using substituted pyrazolo [1,5-a] pyrimidines TYMP, DPYD, TYMS EGLN2 2757/4885FYN 960/4885PDE4D 1156/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.