SCHEMBL11470960

SCHEMBL11470960

NC(=O)c1ccc(-c2nc(C(N)=O)c(O)[nH]2)cc1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 14/20 0.48
IKBKB O14920 1/20 0.46
PKN1 Q16512 1/20 0.44
PKN2 Q16513 1/20 0.44
MKNK1 Q9BUB5 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43
PARP1 P09874 1/20 0.43
RIPK1 Q13546 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11481920 0.90 PARP1 (0.53) CHEK2ADORA2AADORA2BPARP1
SCHEMBL11481631 0.88 PARP1 (0.52) CHEK2ADORA2AADORA2BPARP1
SCHEMBL11485417 0.85 PARP1 (0.52) CHEK2IKBKBPARP1
SCHEMBL11473195 0.85 CHEK2 (0.46) CHEK2PKN1PKN2PARP1
SCHEMBL11473953 0.85 CHEK2 (0.51) CHEK2PARP1
SCHEMBL11474673 0.85 CHEK2 (0.52) CHEK2IKBKBPARP1
SCHEMBL11479983 0.85 PIN1 (0.56) CHEK2IKBKBPARP1
SCHEMBL11472312 0.83 PKN1 (0.51) CHEK2PKN1PKN2MKNK2PARP1
SCHEMBL11472418 0.82 PARP1 (0.60) CHEK2PKN1PKN2PARP1
SCHEMBL11470177 0.81 PARP1 (0.55) CHEK2IKBKBPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4218457-A ANTICANCER ACTIVITY AND IMMUNOSTIMULATING ACTIVITY SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1980-08-19 US disclosed