SCHEMBL1147435

SCHEMBL1147435

CC(C)(C)OC(=O)N[C@](CC=Cc1cccc(Br)c1)(C(=O)O)C1CCCC1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
CTSB P07858 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
SLC6A19 Q695T7 1/20 0.37
NR1H4 Q96RI1 4/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
AAK1 Q2M2I8 3/20 0.35
HSD17B3 P37058 1/20 0.35
BACE1 P56817 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CACNA1B Q00975 1/20 0.34
PKM P14618 1/20 0.34
USP30 Q70CQ3 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1147434 1.00 ALDH1A1 (0.41) ALDH1A1CTSBCTSSCTSKSLC6A19
SCHEMBL490921 0.88 NPC1 (0.42) ALDH1A1CTSSCTSKNR1H4AAK1
SCHEMBL1147485 0.84 AAK1 (0.40) ALDH1A1CTSBCTSSCTSKNR1H4
SCHEMBL1148192 0.78 IKBKB (0.46)
SCHEMBL490801 0.76 AAK1 (0.44) ALDH1A1NR1H4AAK1BACE1KMT2A
SCHEMBL490391 0.76 AAK1 (0.44) ALDH1A1NR1H4AAK1BACE1KMT2A
SCHEMBL490479 0.76 AAK1 (0.39) NR1H4AAK1KMT2AL3MBTL1USP30
SCHEMBL490602 0.74 CHEK1 (0.47) KMT2A
SCHEMBL375738 0.74 EPHX1 (0.38) ALDH1A1CTSSCTSKMAPTKMT2A
SCHEMBL1147982 0.74 CACNA1B (0.53) ALDH1A1CTSBCTSSCTSKSLC6A19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110039920-A1 INHIBITORS OF IKK-BETA SERINE-THERONINE PROTEIN KINASE CHROMA THERAPEUTICS LTD. (GB) 2011-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110039920-A1 INHIBITORS OF IKK-BETA SERINE-THERONINE PROTEIN KINASE CSNK1E, PACSIN2, CHUK ALDH1A1 4456/4885CTSB 974/4885CTSS 1123/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.