SCHEMBL11474686

SCHEMBL11474686

CC(=O)Nc1csc(Cl)n1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.45
KMT2A Q03164 2/20 0.45
PTK2 Q05397 1/20 0.44
ABL1 P00519 5/20 0.44
ADORA3 P0DMS8 4/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
ADORA2A P29274 3/20 0.43
KDM4E B2RXH2 2/20 0.42
MAPT P10636 1/20 0.42
HSD17B10 Q99714 1/20 0.42
LMNA P02545 2/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
DYRK1A Q13627 1/20 0.41
FSCN1 Q16658 1/20 0.41
ADORA1 P30542 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11476352 0.84 P2RY1 (0.44) KMT2AL3MBTL1MEN1RAB9A
SCHEMBL15596971 0.81 NPC1 (0.38) SMN1; SMN2KMT2AMEN1NPC1
SCHEMBL11358850 0.78 L3MBTL1 (0.48) SMN1; SMN2KMT2APTK2ABL1ADORA3
SCHEMBL2642653 0.78 GRM5 (0.44) SMN1; SMN2KMT2AADORA3L3MBTL1ADORA2A
SCHEMBL11350463 0.78 L3MBTL1 (0.62) SMN1; SMN2KMT2AABL1L3MBTL1KDM4E
SCHEMBL2642974 0.77 L3MBTL1 (0.43) SMN1; SMN2KMT2APTK2ABL1ADORA3
SCHEMBL2642609 0.77 PIK3CG (0.53) SMN1; SMN2KMT2AABL1ADORA3L3MBTL1
SCHEMBL2642652 0.77 L3MBTL1 (0.43) SMN1; SMN2KMT2APTK2ABL1ADORA3
SCHEMBL2642608 0.77 L3MBTL1 (0.43) SMN1; SMN2KMT2APTK2ABL1ADORA3
SCHEMBL2642976 0.77 L3MBTL1 (0.43) SMN1; SMN2KMT2APTK2ABL1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4148904-A 2-HALO-4-CARBOXAMIDE- OR CARBOXIMIDOTHIAZOLES JOHN WYETH & BROTHER LIMITED (GB) 1979-04-10 US claimed
CN-102964312-A 4-tertiary butyl-5-(1-aryl-2-nitre ethyl)-2-acylamino thiazole as well as preparation method and application thereof UNIV HUNAN 2013-03-13 CN disclosed
CN-102942536-A 4-tertiary butyl-5-(1-aryl-2-ethyl nitrate)-2-amido-thiazole with insecticidal activity and preparation method thereof UNIV HUNAN 2013-02-27 CN disclosed
CN-102936229-A 4-tertiary butyl-5-benzyl-2-acetyl aminothiazole with insecticidal activity and preparation method UNIV HUNAN 2013-02-20 CN disclosed
US-4183854-A ANTIULCER OR ANTISECRETORY AGENT FOR MAMMALS JOHN WYETH & BROTHER LIMITED (GB) 1980-01-15 US disclosed
US-4148904-A 2-HALO-4-CARBOXAMIDE- OR CARBOXIMIDOTHIAZOLES JOHN WYETH & BROTHER LIMITED (GB) 1979-04-10 US disclosed