SCHEMBL11486308

SCHEMBL11486308

COc1cccc(-c2ccccc2C2=NC(C)(C)CO2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
BACE1 P56817 3/20 0.44
KCNH2 Q12809 2/20 0.44
TDO2 P48775 1/20 0.43
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
NCOA1 Q15788 1/20 0.41
NCOA3 Q9Y6Q9 1/20 0.41
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
DYRK1A Q13627 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1996001 0.88 KDM4E (0.51) KDM4EBACE1KCNH2NCOA1NCOA3
SCHEMBL7112634 0.81 KDM4E (0.53) KDM4EHRH3
SCHEMBL11493291 0.81 KDM4E (0.48) KDM4ENPC1TP53RAB9ASMN1; SMN2
SCHEMBL7571712 0.81 PTPN1 (0.44) KDM4ENPC1TP53NFKB1RAB9A
SCHEMBL11500095 0.80 KDM4E (0.40) KDM4EBACE1NPC1RAB9ASMN1; SMN2
SCHEMBL18380643 0.80 KDM4E (0.61) KDM4EHRH3
SCHEMBL29616919 0.80 KDM4E (0.61) KDM4EHRH3
SCHEMBL7824728 0.79 NPC1 (0.47) KDM4ENPC1RAB9A
SCHEMBL10835648 0.79 KDM4E (0.50) KDM4EHRH3
SCHEMBL8443277 0.78 CYP1A1 (0.56) KDM4EBACE1KCNH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4220778-A ANTIARRHYTHMIC, ANTIMICROBIAL AND CENTRAL NERVOUS SYSTEM ACTIVITY G. D. SEARLE & CO. (US) 1980-09-02 US disclosed