SCHEMBL11488563

SCHEMBL11488563

CCCCNc1nc(N)c2ncn(C3CCCCC3)c2n1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.53
ADORA2A P29274 4/20 0.50
PI4KA P42356 3/20 0.50
PI4K2B Q8TCG2 3/20 0.50
PI4K2A Q9BTU6 3/20 0.50
PI4KB Q9UBF8 3/20 0.50
ADORA2B P29275 1/20 0.50
FLT3 P36888 4/20 0.49
SRC P12931 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
ADORA1 P30542 2/20 0.48
ADORA3 P0DMS8 1/20 0.48
TMIGD3 P0DMS9 1/20 0.47
CDK1 P06493 1/20 0.47
CDK2 P24941 1/20 0.47
PDGFRA P16234 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11489576 0.93 ADORA2A (0.52) CTSLADORA2API4KAPI4K2BPI4K2A
SCHEMBL3125120 0.84 TP53 (0.50) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL12157544 0.81 TP53 (0.49) CTSLADORA2API4KAPI4K2BPI4K2A
SCHEMBL11488562 0.80 ADORA2A (0.50) CTSLADORA2API4KAPI4K2BPI4K2A
SCHEMBL11360463 0.79 ADORA2A (0.57) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL11488384 0.78 ADORA2A (0.60) CTSLADORA2API4KAPI4K2BPI4K2A
SCHEMBL11457082 0.78 ADORA2A (0.58) CTSLADORA2API4KAPI4K2BPI4K2A
SCHEMBL11454848 0.77 ADORA2A (0.58) CTSLADORA2API4KAPI4K2BPI4K2A
SCHEMBL6817943 0.76 CDK2 (0.74) FLT3SRCCDK1CDK2PDGFRA
SCHEMBL6817936 0.76 CDK2 (0.74) FLT3SRCCDK1CDK2PDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3336089-A1 PURINE DERIVATIVES FOR USE IN THE TREATMENT OF ALLERGIC, INFLAMMATORY AND INFECTIOUS DISEASES GlaxoSmithKline LLC (US) 2018-06-20 EP disclosed
US-4232155-A NONADRENERGIC BRONCHODILATOR AGENTS BRISTOL-MYERS COMPANY (US) 1980-11-04 US disclosed