SCHEMBL11489883

SCHEMBL11489883

O=C(OC1C2=C(OCCS2)C(=O)N1c1ccc2ccc(Cl)nc2n1)N1CCNCC1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.34
MAPT P10636 1/20 0.34
RECQL P46063 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRA3 P34903 1/20 0.34
GABRA2 P47869 1/20 0.34
GABRB2 P47870 1/20 0.34
GABRA4 P48169 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11668684 0.90 ADORA3 (0.44) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11484269 0.89 TSHR (0.37) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11493510 0.89 ADORA3 (0.34) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11493503 0.89 ADORA3 (0.34) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11496387 0.89 ADORA3 (0.34) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11493714 0.88 TSHR (0.36) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11486374 0.86 ADORA3 (0.34) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11669036 0.86 ADORA3 (0.34) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11669108 0.81 ADORA3 (0.43) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11492314 0.81 PIK3CD (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4220646-A TRANQUILIZERS, ANTICONVULSANTS, MUSCLE RELAXANTS, HYPNOTIC AGENTS RHONE-POULENC INDUSTRIES (FR) 1980-09-02 US disclosed