SCHEMBL11495271

SCHEMBL11495271

CN(C)Cc1c(Cc2ccccc2)[nH]c2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.61
MAPT P10636 4/20 0.61
TSHR P16473 4/20 0.54
CYP2C19 P33261 4/20 0.54
CYP1A2 P05177 3/20 0.54
HPGD P15428 3/20 0.54
TDP1 Q9NUW8 3/20 0.54
MTNR1A P48039 2/20 0.54
MTNR1B P49286 2/20 0.54
CYP2C9 P11712 2/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
HTR6 P50406 1/20 0.49
ALDH1A1 P00352 5/20 0.48
CYP2D6 P10635 3/20 0.48
ALOX15 P16050 1/20 0.48
HSD17B10 Q99714 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11493601 0.86 MAPT (0.52) CYP3A4MAPTTSHRCYP2C19CYP1A2
SCHEMBL31034424 0.83 HPGD (0.58) CYP3A4MAPTTSHRCYP2C19CYP1A2
SCHEMBL18919603 0.79 TSHR (0.58) CYP3A4MAPTTSHRCYP2C19CYP1A2
SCHEMBL11495550 0.77 CYP3A4 (0.52) CYP3A4MAPTTSHRCYP2C19MEN1
SCHEMBL14540350 0.77 CYP3A4 (0.64) CYP3A4MAPTTSHRCYP2C19MEN1
2-Methyl Gramine SCHEMBL2519973 0.76 MAPT (1.00) CYP3A4MAPTTSHRCYP2C19CYP1A2
SCHEMBL8804026 0.76 MTNR1A (0.59) CYP3A4MAPTTSHRCYP2C19CYP1A2
SCHEMBL11495830 0.76 HTR2A (0.71) CYP3A4MAPTCYP2C19CYP1A2HPGD
SCHEMBL2087168 0.75 HPGD (0.61) CYP3A4MAPTTSHRCYP2C19CYP1A2
SCHEMBL28543275 0.75 AHR (0.52) CYP3A4MAPTTSHRCYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4217357-A Inhibition of thromboxane synthetase with 3-(imidazol-1-ylalkyl)indoles PFIZER INC. (US) 1980-08-12 US disclosed