SCHEMBL11503528

SCHEMBL11503528

C#CC[C@H](CCCC)OC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.33
PRSS1 P07477 1/20 0.31
CTSG P08311 1/20 0.31
CTRB1 P17538 1/20 0.31
CMA1 P23946 1/20 0.31
KIF11 P52732 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
TSHR P16473 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11340509 1.00 CNR2 (0.33) CNR2PRSS1CTSGCTRB1CMA1
SCHEMBL11346882 0.84 KIF11 (0.33) KIF11CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL11730456 0.80 CNR2 (0.35) CNR2PRSS1CTSGCTRB1CMA1
SCHEMBL11503551 0.78 KIF11 (0.31) KIF11
SCHEMBL10682475 0.76 CNR2 (0.36) CNR2PRSS1CTSGCTRB1CMA1
SCHEMBL11561124 0.75 CNR2 (0.35) CNR2PRSS1CTSGCTRB1CMA1
SCHEMBL11107646 0.75 CSNK1E (0.36) CNR2PRSS1CTSGCTRB1CMA1
SCHEMBL11107718 0.75 CSNK1E (0.36) CNR2PRSS1CTSGCTRB1CMA1
SCHEMBL11503682 0.74 KIF11 (0.35) KIF11CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL11503776 0.74 CNR2 (0.31) CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4179451-A HYPOTENSIVE, ANTIULCER, BRONCHODILATOR, ANTICONVULSANTS OR ANTIMICROBIAL AGENTS AMERICAN CYANAMID COMPANY (US) 1979-12-18 US disclosed
US-4107441-A HYPOTENSIVE, ANTIULCER, BRONCHODILATORS, ANTIMICROBIAL, ANTICONVULSANTS AMERICAN CYANAMID COMPANY (US) 1978-08-15 US disclosed
US-4061672-A Derivatives of 9-hydroxy-13-trans-prostenoic acid AMERICAN CYANAMID COMPANY (US) 1977-12-06 US disclosed
US-RE29469-E PROSTAGLANDINS; BRONCHODILATORS, HYPOTENSIVES, ANTIULCER AGENTS AMERICAN CYANAMID COMPANY (US) 1977-11-08 US disclosed
US-3950406-A BRONCHODILATORS, HYPOTENSIVE, ANTIULCER AMERICAN CYANAMID COMPANY (US) 1976-04-13 US disclosed