SCHEMBL11514768

SCHEMBL11514768

CCOC(=O)C(=CNc1ccnc(-c2cccnc2)n1)C(=O)OCC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 8/20 0.56
KMT2A Q03164 4/20 0.56
MEN1 O00255 1/20 0.56
MAPT P10636 4/20 0.54
KDM4E B2RXH2 1/20 0.54
CYP3A4 P08684 6/20 0.53
CYP2C19 P33261 6/20 0.53
CYP2C9 P11712 4/20 0.53
CYP2D6 P10635 6/20 0.52
MAPK1 P28482 2/20 0.52
HTT P42858 1/20 0.52
NPSR1 Q6W5P4 1/20 0.51
IDE P14735 1/20 0.51
CLK4 Q9HAZ1 4/20 0.50
ALDH1A1 P00352 2/20 0.49
POLB P06746 1/20 0.49
TDP1 Q9NUW8 2/20 0.49
PPARG P37231 1/20 0.49
NR2E3 Q9Y5X4 1/20 0.49
NCOR2 Q9Y618 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11515727 0.86 MEN1 (0.57) CYP1A2KMT2AMEN1MAPTKDM4E
SCHEMBL11648801 0.83 MEN1 (0.59) CYP1A2KMT2AMEN1MAPTKDM4E
SCHEMBL11515259 0.83 CYP1A2 (0.61) CYP1A2KMT2AMEN1MAPTKDM4E
SCHEMBL11651691 0.83 MEN1 (0.53) CYP1A2KMT2AMEN1MAPTKDM4E
SCHEMBL11651088 0.82 MEN1 (0.58) CYP1A2KMT2AMEN1MAPTKDM4E
SCHEMBL11517088 0.81 MEN1 (0.51) CYP1A2KMT2AMEN1MAPTKDM4E
SCHEMBL11517093 0.81 MEN1 (0.51) CYP1A2KMT2AMEN1MAPTKDM4E
SCHEMBL11514663 0.80 MAPT (0.51) CYP1A2KMT2AMEN1MAPTKDM4E
SCHEMBL11514659 0.80 MAPT (0.51) CYP1A2KMT2AMEN1MAPTKDM4E
SCHEMBL11652035 0.80 MAPT (0.54) CYP1A2KMT2AMEN1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE30024-E ANTIALLERGENS STERLING DRUG INC. (US) 1979-06-05 US disclosed
US-4118571-A ANTIALLERGENS STERLING DRUG INC. (US) 1978-10-03 US disclosed
US-4086233-A ANTIALLERGENS STERLING DRUG INC. (US) 1978-04-25 US disclosed
US-4032523-A ANTIALLERGENS STERLING DRUG INC. (US) 1977-06-28 US disclosed
US-4018770-A ANTIALLERGENS STERLING DRUG INC. (US) 1977-04-19 US disclosed
US-3992380-A 5,8-Dihydro-5-oxo-2-(4-or 3-pyridinyl)pyrido[2,3-d]pyrimidine-6-carboxylic acids and esters STERLING DRUG INC. (US) 1976-11-16 US disclosed