SCHEMBL11515740

SCHEMBL11515740

C[CH]CCc1cnccn1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
XDH P47989 1/20 0.32
TXNRD1 Q16881 1/20 0.32
HRH1 P35367 6/20 0.32
CYP2D6 P10635 5/20 0.32
KCNH2 Q12809 2/20 0.32
CHRM1 P11229 1/20 0.32
HTR2A P28223 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRA5 P31644 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27866178 0.80 HRH1 (0.33) HSP90AA1PDCD1CD274CYP1A2CYP3A4
SCHEMBL1778280 0.79 HSP90AA1 (0.33) HSP90AA1PDCD1CD274CYP1A2CYP3A4
SCHEMBL3301973 0.79 HDAC3 (0.36) HSP90AA1PDCD1CD274CYP1A2CYP3A4
SCHEMBL30390174 0.76
SCHEMBL309452 0.76
SCHEMBL1829926 0.75 ALDH1A1 (0.38) HSP90AA1PDCD1CD274CYP1A2CYP3A4
SCHEMBL28362525 0.75 HSP90AA1 (0.40) HSP90AA1CYP1A2CYP3A4HDAC3HDAC1
Ethane SCHEMBL28701355 0.74 CYP3A4 (0.39) HSP90AA1CYP1A2CYP3A4HDAC3HDAC1
Ethane SCHEMBL29272596 0.72 HRH1 (0.35) HSP90AA1PDCD1CD274CYP1A2CYP3A4
SCHEMBL4412197 0.72 CYP2D6 (0.43) CYP3A4CYP2C9CYP2C19HRH1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4138410-A Flavoring agent FIRMENICH & CIE (CH) 1979-02-06 US disclosed
US-4126618-A FLAVOR ADDITIVES FOR FOODS AND BEVERAGES FIRMENICH & CIE (CH) 1978-11-21 US disclosed
US-3989713-A Pyrrylmethylthio flavoring agents FIRMENICH & CIE (CH) 1976-11-02 US disclosed
US-3952026-A FLAVOR ADDITIVE FOR FOODS AND BEVERAGES FIRMENICH & CIE (CH) 1976-04-20 US disclosed
US-3952024-A FLAVOR ADDITIVE FOR FOODS AND BEVERAGES FIRMENICH & CIE (CH) 1976-04-20 US disclosed
US-3943260-A TETRAHYDRO-THIO-PHEN-3-ONES FIRMENICH & CIE (CH) 1976-03-09 US disclosed
US-3931166-A FLAVORANTS FIRMENICH & CIE (CH) 1976-01-06 US disclosed
US-3931246-A FURYLALKYL-THIOETHERS FIRMENICH & CIE (CH) 1976-01-06 US disclosed
US-3931245-A FURYLALKYLTHIOL CARBOXYLATES FIRMENICH & CIE (CH) 1976-01-06 US disclosed