SCHEMBL11525975

SCHEMBL11525975

O=C(O)CCc1nnn(Cc2ccccc2)c1O

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.50
HPGD P15428 1/20 0.48
KEAP1 Q14145 1/20 0.47
CYP2C19 P33261 1/20 0.47
POLB P06746 1/20 0.47
FFAR1 O14842 1/20 0.45
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HTT P42858 1/20 0.44
IDO1 P14902 1/20 0.44
HCAR3 P49019 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
TSHR P16473 1/20 0.43
SLC9A1 P19634 1/20 0.43
GRM2 Q14416 1/20 0.43
HSD11B1 P28845 1/20 0.43
CYP1A2 P05177 1/20 0.43
EGLN3 Q9H6Z9 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11530977 0.84 GAA (0.49) GAAHPGDKEAP1CYP2C19POLB
SCHEMBL11534274 0.83 CYP19A1 (0.51) POLBKDM4EALDH1A1SMN1; SMN2CYP1A2
SCHEMBL11534999 0.83 GAA (0.48) GAAHPGDKEAP1CYP2C19POLB
SCHEMBL15875517 0.75 HPGD (0.69) GAAHPGDALDH1A1HTTIDO1
SCHEMBL9477798 0.75 HDAC1 (0.52) GAAKEAP1ALDH1A1TSHRHSD11B1
SCHEMBL17286362 0.73 HPGD (0.61) GAAHPGDCYP2C19ALDH1A1HTT
SCHEMBL17283076 0.73 HPGD (0.57) GAAHPGDALDH1A1HTTIDO1
SCHEMBL11535000 0.72 HDAC3 (0.44) GAAHPGDCYP2C19POLBALDH1A1
SCHEMBL21606708 0.72 HSD11B1 (0.77) GAAHPGDKEAP1FFAR1SMN1; SMN2
SCHEMBL11528186 0.70 CYP19A1 (0.51) POLBKDM4EALDH1A1SMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4142046-A BACTERICIDES, 7-AMINO-CEPHALOSPORINS SMITHKLINE CORPORATION (US) 1979-02-27 US disclosed
US-4060610-A Pharmaceutical compositions comprising 7-acyl-3-(substituted triazolyl thiomethyl)-cephalosporins and methods of treating bacterial infections SMITHKLINE CORPORATION (US) 1977-11-29 US disclosed
US-3989694-A ANTIBACTERIAL SMITHKLINE CORPORATION (US) 1976-11-02 US disclosed