SCHEMBL11528161

SCHEMBL11528161

Cc1ccc2c(c1)Nc1cscc1C(N1CCN(C)CC1)=N2

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 6/20 0.52
DRD2 P14416 6/20 0.52
HRH4 Q9H3N8 2/20 0.52
NFKB1 P19838 2/20 0.51
BLM P54132 2/20 0.51
NPSR1 Q6W5P4 1/20 0.51
CHRM1 P11229 8/20 0.50
HRH1 P35367 4/20 0.50
DRD3 P35462 3/20 0.50
CHRM2 P08172 3/20 0.50
CHRM4 P08173 3/20 0.50
CHRM5 P08912 3/20 0.50
ADRA2A P08913 3/20 0.50
ADRA2B P18089 3/20 0.50
ADRA2C P18825 3/20 0.50
CHRM3 P20309 3/20 0.50
DRD1 P21728 3/20 0.50
ADRA1D P25100 3/20 0.50
HTR2A P28223 3/20 0.50
HTR2C P28335 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11666986 0.91 CHRM1 (0.57) DRD4DRD2HRH4NFKB1BLM
SCHEMBL11531362 0.87 CHRM1 (0.62) DRD4DRD2HRH4CHRM1HRH1
SCHEMBL11633189 0.87 DRD2 (0.61) DRD4DRD2HRH4NFKB1BLM
SCHEMBL11631048 0.87 CHRM1 (0.61) DRD4DRD2HRH4NFKB1BLM
SCHEMBL11631603 0.85 DRD2 (0.49) DRD4DRD2HRH4NFKB1BLM
SCHEMBL11634162 0.85 CHRM1 (0.63) DRD4DRD2HRH4NFKB1BLM
SCHEMBL11531378 0.84 DRD2 (0.74) DRD4DRD2HRH4NFKB1BLM
SCHEMBL11534075 0.82 CHRM1 (0.52) DRD4DRD2HRH4NFKB1BLM
SCHEMBL11529616 0.82 CHRM1 (0.55) DRD4DRD2HRH4NFKB1BLM
SCHEMBL11632479 0.81 CHRM1 (0.71) DRD4DRD2HRH4NFKB1BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4172831-A CENTRAL NERVOUS SYSTEM LILLY INDUSTRIES LIMITED (GB) 1979-10-30 US disclosed
US-4115574-A CNS ACTIVITY LILLY INDUSTRIES LIMITED (GB) 1978-09-19 US disclosed
US-4115568-A CNS ACTIVITY LILLY INDUSTRIES LIMITED (GB) 1978-09-19 US disclosed