SCHEMBL11530499

SCHEMBL11530499

CCc1cc2c(s1)C(N1CCN(C)CC1)=Nc1cc(Cl)ccc1N2

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.60
DRD4 P21917 6/20 0.60
CHRM1 P11229 4/20 0.60
HRH4 Q9H3N8 4/20 0.60
DRD3 P35462 3/20 0.60
HRH1 P35367 2/20 0.60
HTR3E A5X5Y0 1/20 0.60
MEN1 O00255 1/20 0.60
CACNA1F O60840 1/20 0.60
HTR3B O95264 1/20 0.60
ABCB11 O95342 1/20 0.60
LMNA P02545 1/20 0.60
CYP1A2 P05177 1/20 0.60
POLB P06746 1/20 0.60
ADRB2 P07550 1/20 0.60
CHRM2 P08172 1/20 0.60
CHRM4 P08173 1/20 0.60
CYP3A4 P08684 1/20 0.60
HTR1A P08908 1/20 0.60
CHRM5 P08912 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11530432 0.87 CHRM1 (0.47) DRD2DRD4CHRM1HRH4DRD3
SCHEMBL11528431 0.87 CHRM1 (0.64) CHRM1HRH1PAK1
SCHEMBL11529453 0.86 CHRM1 (0.64) DRD2DRD4CHRM1HRH4DRD3
SCHEMBL11531565 0.86 DRD2 (0.59) DRD2DRD4CHRM1HRH4DRD3
SCHEMBL11533782 0.85 CHRM1 (0.47) DRD2DRD4CHRM1HRH4DRD3
SCHEMBL11531705 0.85 CHRM1 (0.45) DRD2DRD4CHRM1HRH4DRD3
SCHEMBL11532957 0.83 CHRM1 (0.43) DRD2DRD4CHRM1HRH4DRD3
SCHEMBL11532641 0.83 CHRM1 (0.46) DRD2CHRM1HRH1CHRM2CHRM4
SCHEMBL11535016 0.82 HRH4 (0.46) DRD2DRD4CHRM1HRH4DRD3
SCHEMBL11532012 0.81 CHRM1 (0.66) DRD2DRD4CHRM1HRH4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4172831-A CENTRAL NERVOUS SYSTEM LILLY INDUSTRIES LIMITED (GB) 1979-10-30 US disclosed
US-4115574-A CNS ACTIVITY LILLY INDUSTRIES LIMITED (GB) 1978-09-19 US disclosed
US-4115568-A CNS ACTIVITY LILLY INDUSTRIES LIMITED (GB) 1978-09-19 US disclosed