SCHEMBL11538360

SCHEMBL11538360

CC(C)NC(=O)c1cccnc1N

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 2/20 0.58
NAPRT Q6XQN6 1/20 0.56
ALOX5 P09917 1/20 0.47
VCP P55072 4/20 0.47
MAPK8 P45983 1/20 0.47
P2RX7 Q99572 1/20 0.46
PDE4A P27815 1/20 0.46
KCNH2 Q12809 1/20 0.46
EIF2S1 P05198 1/20 0.44
EIF2AK3 Q9NZJ5 1/20 0.44
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
RIPK1 Q13546 1/20 0.43
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19090781 0.84 PRKCI (0.55) PRKCINAPRTVCPP2RX7ALDH1A1
SCHEMBL165047 0.81 MAPK8 (0.48) ALOX5MAPK8P2RX7PDE4AKCNH2
SCHEMBL268777 0.81 P2RX7 (0.65) MAPK8P2RX7PDE4AKCNH2ALDH1A1
SCHEMBL26336039 0.81 MAPK8 (0.48) ALOX5MAPK8P2RX7PDE4AKCNH2
SCHEMBL1232303 0.81 PRKCI (0.63) PRKCINAPRTVCPP2RX7LMNA
SCHEMBL27559774 0.81 KDM4E (0.46) ALOX5MAPK8P2RX7PDE4AKCNH2
SCHEMBL24571401 0.80 SMN1; SMN2 (0.56) ALDH1A1LMNAMAPTHPGDSMN1; SMN2
SCHEMBL27986290 0.80 MAPK8 (0.47) MAPK8P2RX7PDE4AKCNH2ALDH1A1
SCHEMBL21209660 0.80 NAPRT (0.56) NAPRTALOX5MAPK8P2RX7PDE4A
SCHEMBL11906279 0.80 KDM4E (0.51) PRKCIMAPK8PDE4AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115969846-B Application of small molecule compound LZ-10 in preparation of medicine for treating and/or preventing optic neuritis lineage diseases 上海中医药大学附属岳阳中西医结合医院 2024-04-12 CN claimed
CN-115969846-A Application of small molecule compound LZ-10 in preparing medicine for treating and/or preventing optic neuritis pedigree diseases 上海中医药大学附属岳阳中西医结合医院 2023-04-18 CN claimed
CN-115969846-B Application of small molecule compound LZ-10 in preparation of medicine for treating and/or preventing optic neuritis lineage diseases 上海中医药大学附属岳阳中西医结合医院 2024-04-12 CN disclosed
CN-115969846-A Application of small molecule compound LZ-10 in preparing medicine for treating and/or preventing optic neuritis pedigree diseases 上海中医药大学附属岳阳中西医结合医院 2023-04-18 CN disclosed
CN-102574845-A 1h-imidazo[4,5-c]quinolinone derivatives NOVARTIS AG 2012-07-11 CN disclosed
US-4175184-A Manufacture of 2,1,3-thiadiazin-4-one-2,2-dioxide derivatives BASF AKTIENGESELLSCHAFT (DE) 1979-11-20 US disclosed
US-3947442-A Method for producing heterocyclic acid anhydrides and pyrimidinediones THE SHERWIN-WILLIAMS COMPANY (US) 1976-03-30 US disclosed
US-3947416-A Azaisatoic anhydrides THE SHERWIN-WILLIAMS COMPANY (US) 1976-03-30 US disclosed