SCHEMBL11540971

SCHEMBL11540971

ClC1=CN2CCN=C2C(Cl)=C1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
GLA P06280 1/20 0.53
GAA P10253 1/20 0.53
PTAFR P25105 3/20 0.33
SMARCA2 P51531 1/20 0.32
HDAC8 Q9BY41 2/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30
HDAC4 P56524 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3851283 0.81 KDM4E (0.39) KDM4EALDH1A1GLAGAA
SCHEMBL20125021 0.81 KDM4E (0.36) KDM4EALDH1A1GLAGAA
SCHEMBL11539073 0.60 KDM4E (0.30) KDM4EALDH1A1GAA
SCHEMBL14309129 0.60 HDAC8 (0.30) HDAC8HDAC4
SCHEMBL8446377 0.59 HDAC8 (0.33) HDAC8HDAC4HDAC6
SCHEMBL11299918 0.56
SCHEMBL14309130 0.56 HRH4 (0.33)
SCHEMBL2606658 0.52 KDM4E (0.51) KDM4EALDH1A1HDAC8
SCHEMBL16041282 0.46
SCHEMBL1316573 0.43 NOS1 (0.40) ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4163745-A ANTIDIABETIC, HYPOGLYCEMIC PFIZER INC. (US) 1979-08-07 US disclosed
US-4141898-A Imidazo pyridinium quaternary salts as hypoglycemic agents PFIZER INC. (US) 1979-02-27 US disclosed
US-4129567-A IMIDAZOPYRIDINES AND ISOB IDINE PFIZER INC. (US) 1978-12-12 US disclosed
US-4093616-A PYRROLO(1,2-A)PYRAZINIUM, PYRAZOLO(1,5-A)PYRIDINIUM, 1H-IMIDAZO(2,1-A)ISOQUINOLINIUM, OR IMIDAZO(5,1-A)ISOQUINOLINIUM SALTS PFIZER INC. (US) 1978-06-06 US disclosed
US-4044015-A Imidazopyridinium compounds as hypoglycemic agents PFIZER INC. (US) 1977-08-23 US disclosed