SCHEMBL11544266

SCHEMBL11544266

Clc1cccc(Cl)c1C1(Cn2cncn2)OCCO1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.46
THRB P10828 1/20 0.46
KDM4E B2RXH2 2/20 0.43
CYP2C9 P11712 3/20 0.42
CYP19A1 P11511 2/20 0.41
HSP90AA1 P07900 3/20 0.40
NPSR1 Q6W5P4 1/20 0.40
GAA P10253 1/20 0.38
HSD17B10 Q99714 1/20 0.38
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
ALDH1A1 P00352 2/20 0.36
KMT2A Q03164 2/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C19 P33261 2/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11543211 0.87 CYP3A4 (0.51) CYP3A4THRBKDM4ECYP2C9CYP19A1
SCHEMBL11544361 0.86 CYP3A4 (0.50) CYP3A4THRBKDM4ECYP2C9CYP19A1
SCHEMBL11542064 0.81 CYP3A4 (0.48) CYP3A4THRBCYP2C9CYP19A1HSP90AA1
SCHEMBL9087421 0.80 CYP3A4 (0.52) CYP3A4THRBKDM4ECYP2C9CYP19A1
SCHEMBL11545660 0.80 CYP3A4 (0.49) CYP3A4THRBKDM4ECYP2C9HSP90AA1
SCHEMBL11545358 0.80 SLC6A4 (0.53) CYP3A4THRBCYP2C9HSP90AA1NPSR1
SCHEMBL9729882 0.79 GAA (0.51) CYP3A4THRBKDM4ECYP2C9CYP19A1
SCHEMBL11540746 0.79 CYP3A4 (0.56) CYP3A4THRBKDM4ECYP2C9HSP90AA1
Azaconazole SCHEMBL29354903 0.79 CYP3A4 (0.69) CYP3A4THRBKDM4ECYP2C9HSP90AA1
Azaconazole SCHEMBL21056 0.79 CYP3A4 (0.69) CYP3A4THRBKDM4ECYP2C9HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4160838-A FUNGICIDES, BACTERICIDES JANSSEN PHARMACEUTICA N.V. (BE) 1979-07-10 US disclosed
US-4079062-A ANTIMICROBIAL, PLANT GROWTH REGULATORS; 1-(B-ARYL)ETHYL-1H-1,2,4-TRIAZOLE KETALS JANSSEN PHARMACEUTICA N.V. (BE) 1978-03-14 US disclosed