Azaconazole

Azaconazole

SCHEMBL21056

Clc1ccc(C2(Cn3cncn3)OCCO2)c(Cl)c1

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 16/20 0.69
THRB P10828 1/20 0.69
CYP2C9 P11712 3/20 0.60
LMNA P02545 2/20 0.49
FYN P06241 2/20 0.49
CYP51A1 Q16850 2/20 0.49
NR1I2 O75469 1/20 0.49
PGR P06401 1/20 0.49
HSP90AA1 P07900 1/20 0.49
CHRM2 P08172 1/20 0.49
CHRM4 P08173 1/20 0.49
CHRM5 P08912 1/20 0.49
ADRA2A P08913 1/20 0.49
CHRM1 P11229 1/20 0.49
TSHR P16473 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
CHRM3 P20309 1/20 0.49
DRD1 P21728 1/20 0.49
TBXA2R P21731 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Azaconazole SCHEMBL3009257 1.00 CYP3A4 (0.69) CYP3A4THRBCYP2C9LMNAFYN
Azaconazole SCHEMBL29354903 1.00 CYP3A4 (0.69) CYP3A4THRBCYP2C9LMNAFYN
Azaconazole SCHEMBL29017725 0.99 CYP3A4 (0.67) CYP3A4THRBCYP2C9LMNAFYN
SCHEMBL2127240 0.95 CYP3A4 (0.66) CYP3A4THRBCYP2C9LMNAFYN
Azaconazole SCHEMBL11544952 0.93 CYP3A4 (0.61) CYP3A4THRBCYP2C9LMNAFYN
Azaconazole SCHEMBL11543267 0.91 KDM4E (0.60) CYP3A4THRBCYP2C9LMNAFYN
SCHEMBL11540746 0.90 CYP3A4 (0.56) CYP3A4THRBCYP2C9LMNAFYN
Azaconazole SCHEMBL10712944 0.89 CYP3A4 (0.57) CYP3A4THRBCYP2C9LMNAFYN
Azaconazole SCHEMBL2364039 0.88 CYP3A4 (0.56) CYP3A4THRBCYP2C9LMNAFYN
SCHEMBL10707904 0.88 CYP3A4 (0.57) CYP3A4THRBCYP2C9LMNAFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 22310 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137082-A1 FUNGICIDAL COMPOSITIONS COMPRISING FLUDIOXONIL SYNGENTA CROP PROTECTION AG (CH) 2026-05-21 US claimed
WO-2026105160-A1 NOVEL AGROCHEMICAL COMPOSITION COMPRISING 3-SUBSTITUTED PHENYLAMIDINE COMPOUNDS AND USE THEREOF PI INDUSTRIES LTD. (IN) 2026-05-21 WO claimed
US-20260101900-A1 OIL LIQUID FUNGICIDAL FORMULATION ADAMA MAKHTESHIM LTD. (IL) 2026-04-16 US claimed
US-20260101893-A1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2026-04-16 US claimed
US-20260076366-A1 SYNERGISTIC PESTICIDAL COMPOSITIONS AND METHODS FOR DELIVERY OF ACTIVE INGREDIENTS 0903608 B C LTD (CA) 2026-03-19 US claimed
US-20260076371-A1 AGROCHEMICAL COMPOSITION OF TRIAZOLES ADAMA MAKHTESHIM LTD. (IL) 2026-03-19 US claimed
EP-4710766-A1 MIXTURES OF AMBRUTICIN WITH AT LEAST ONE FURTHER PESTICIDE BASF SE (DE) 2026-03-18 EP claimed
US-20260068884-A1 COMPOSITION USED FOR KILLING FUNGI AND METHOD FOR APPLYING COMPOSITION JIANGSU FLAG CHEMICAL INDUSTRY CO., LTD. (CN) 2026-03-12 US claimed
WO-2026041871-A1 METHODS OF CONTROLLING CAUSAL AGENTS OF RAMULARIA LEAF SPOT OR RHYNCHOSPORIUM LEAF SCALD DISEASE, AND COMPOSITIONS FOR THE SAME GOWAN CROP PROTECTION LIMITED (GB) 2026-02-26 WO claimed
EP-4114183-B1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2026-02-25 EP claimed
EP-0148526-B1 WATER-DILUTABLE WOOD-PRESERVING LIQUIDS JANSSEN PHARMACEUTICA N.V. (BE) 1988-04-27 EP claimed
EP-0101102-B1 PREVENTING FUNGAL DECAY OF FOOD PRODUCTS, PARTICULARLY HARVESTED FRUITS JANSSEN PHARMACEUTICA N.V. (BE) 1988-04-06 EP claimed
EP-0252875-A2 Microbicidal agent CIBA-GEIGY AG (CH) 1988-01-13 EP claimed
US-4648988-A AZOLE, SOLVENT, SOLUBILIZER JANSSEN PHARMACEUTICA, N.V. (BE) 1987-03-10 US claimed
US-4542146-A Process for the protection of wood and coatings against deterioration by microorganisms JANSSEN PHARMACEUTICA N.V. (BE) 1985-09-17 US claimed
EP-0148526-A1 Water-dilutable wood-preserving liquids JANSSEN PHARMACEUTICA N.V. (BE) 1985-07-17 EP claimed
EP-0038109-B1 AGENTS AND METHOD FOR THE PROTECTION OF COATINGS AND WOOD AND OTHER NON-LIVING ORGANIC SUBSTRATES FROM DETERIORATION BY MICRO-ORGANISMS JANSSEN PHARMACEUTICA N.V. (BE) 1984-08-29 EP claimed
EP-0101102-A2 Preventing fungal decay of food products, particularly harvested fruits JANSSEN PHARMACEUTICA N.V. (BE) 1984-02-22 EP claimed
US-4160838-A FUNGICIDES, BACTERICIDES JANSSEN PHARMACEUTICA N.V. (BE) 1979-07-10 US claimed
US-4079062-A ANTIMICROBIAL, PLANT GROWTH REGULATORS; 1-(B-ARYL)ETHYL-1H-1,2,4-TRIAZOLE KETALS JANSSEN PHARMACEUTICA N.V. (BE) 1978-03-14 US claimed