SCHEMBL11545733

SCHEMBL11545733

COc1ccc(C(O)CNCCc2ccc(OC)c(OC)c2)cc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 10/20 0.81
ADRB1 P08588 6/20 0.81
SLC6A4 P31645 2/20 0.81
SLC6A3 Q01959 2/20 0.81
ALDH1A1 P00352 1/20 0.81
LMNA P02545 1/20 0.81
NPSR1 Q6W5P4 1/20 0.81
SLC22A1 O15245 1/20 0.81
CHRM2 P08172 1/20 0.81
CYP3A4 P08684 1/20 0.81
CHRM1 P11229 1/20 0.81
TSHR P16473 1/20 0.81
NFKB1 P19838 1/20 0.81
OPRM1 P35372 1/20 0.81
HIF1A Q16665 1/20 0.81
ADRB3 P13945 4/20 0.63
KDM4E B2RXH2 2/20 0.62
GAA P10253 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
TDP1 Q9NUW8 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10718998 0.90 ADRB2 (0.67) ADRB2ADRB1SLC6A4SLC6A3ALDH1A1
Denopamine SCHEMBL218640 0.90 ADRB2 (1.00) ADRB2ADRB1SLC6A4SLC6A3ALDH1A1
Denopamine SCHEMBL29964546 0.90 ADRB2 (1.00) ADRB2ADRB1SLC6A4SLC6A3ALDH1A1
SCHEMBL11710152 0.90 ADRB2 (0.81) ADRB2ADRB1SLC6A4SLC6A3ALDH1A1
Denopamine SCHEMBL218641 0.90 ADRB2 (1.00) ADRB2ADRB1SLC6A4SLC6A3ALDH1A1
Denopamine SCHEMBL4542605 0.90 ADRB2 (1.00) ADRB2ADRB1SLC6A4SLC6A3ALDH1A1
SCHEMBL10720260 0.89 ADRB2 (0.65) ADRB2ADRB1SLC6A4SLC6A3ALDH1A1
Denopamine SCHEMBL7338329 0.89 ADRB2 (0.97) ADRB2ADRB1SLC6A4SLC6A3ALDH1A1
SCHEMBL11257835 0.88 ADRB2 (1.00) ADRB2ADRB1SLC6A4SLC6A3ALDH1A1
Hydrochloric Acid SCHEMBL11710346 0.88 ADRB2 (0.78) ADRB2ADRB1SLC6A4SLC6A3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4172890-A CARDIOVASCULAR, PARKINSON'S DISEASE, DOPAMINERGIC SMITHKLINE CORPORATION (US) 1979-10-30 US disclosed
US-4108989-A TREATING PARKINSON*S DISEASE, CARDIOVASCULAR DISORDERS SMITHKLINE CORPORATION (US) 1978-08-22 US disclosed
US-4011319-A STIMULATING DOPAMINE RECEPTORS, RENAL VASODILATORS, DIURETICS SMITHKLINE CORPORATION (US) 1977-03-08 US disclosed