SCHEMBL11547740

SCHEMBL11547740

CCOC(=O)CC(C)(O)c1ccc(Oc2ccc(Cl)cc2)cc1F

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
ABCB11 O95342 1/20 0.43
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43
HTR2A P28223 1/20 0.43
PMP22 Q01453 1/20 0.43
PPARA Q07869 1/20 0.43
OPRK1 P41145 1/20 0.38
ALDH1A1 P00352 1/20 0.37
MAPK14 Q16539 1/20 0.37
P2RX3 P56373 3/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
MAPT P10636 1/20 0.36
POLB P06746 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
ALOX5 P09917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11543977 0.87 PTGDR2 (0.40) CYP1A2CYP3A4PPARAMAPK14P2RX3
SCHEMBL11507387 0.81 CYP1A2 (0.50) CYP1A2ABCB11CYP3A4TSHRHTR2A
SCHEMBL31294683 0.80 MAPT (0.41) CYP1A2CYP3A4TSHRALDH1A1MAPT
SCHEMBL11544106 0.79 MAOA (0.39) CYP1A2ABCB11CYP3A4TSHRHTR2A
SCHEMBL11546454 0.78 MAPK14 (0.38) CYP3A4HTR2APPARAMAPK14MAOA
SCHEMBL11547739 0.77 SCN9A (0.41) CYP1A2ABCB11CYP3A4TSHRHTR2A
SCHEMBL22439742 0.76 PPARA (0.45) CYP1A2CYP3A4PPARAMAPK14MAOA
SCHEMBL11506945 0.75 CYP2C9 (0.44) CYP1A2ABCB11CYP3A4TSHRHTR2A
SCHEMBL21991523 0.75 PPARA (0.58) CYP1A2ABCB11CYP3A4TSHRHTR2A
SCHEMBL22407020 0.74 MAPK14 (0.40) CYP1A2ABCB11CYP3A4TSHRHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4151302-A Araliphatic dihalogen compounds composition and method of use MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-04-24 US disclosed
US-4057647-A Araliphatic dihalogen compounds and process for their preparation MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-11-08 US disclosed