SCHEMBL11550353

SCHEMBL11550353

CCCCOC(=O)C=C(N)N(C)C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.55
TSHR P16473 3/20 0.52
HPGD P15428 2/20 0.52
RAB9A P51151 3/20 0.50
MAPT P10636 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
HCAR2 Q8TDS4 4/20 0.49
ALDH1A1 P00352 4/20 0.44
APP P05067 1/20 0.37
ESR1 P03372 1/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
PDE4D Q08499 1/20 0.37
NAAA Q02083 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NPC1 O15118 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11550350 1.00 ATM (0.55) ATMTSHRHPGDRAB9AMAPT
SCHEMBL11563279 1.00 ATM (0.55) ATMTSHRHPGDRAB9AMAPT
SCHEMBL11563575 0.81 ATM (0.63) ATMTSHRHPGDRAB9AMAPT
SCHEMBL11555877 0.81 NPSR1 (0.50) TSHRMAPTNPSR1HCAR2ALDH1A1
SCHEMBL11548834 0.81 NPSR1 (0.50) TSHRMAPTNPSR1HCAR2ALDH1A1
SCHEMBL11548836 0.81 NPSR1 (0.50) TSHRMAPTNPSR1HCAR2ALDH1A1
SCHEMBL11567146 0.80 CHRM1 (0.52) MAPTNPSR1ALDH1A1LMNACYP1A2
SCHEMBL11560554 0.80 SMN1; SMN2 (0.36) ATMTSHRRAB9AMAPTNPSR1
SCHEMBL11567144 0.80 CHRM1 (0.52) MAPTNPSR1ALDH1A1LMNACYP1A2
SCHEMBL11560557 0.80 SMN1; SMN2 (0.36) ATMTSHRRAB9AMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4162321-A Sulphur-containing amino-dihydropyridines, and their use as medicants BAYER AKTIENGESELLSCHAFT (DE) 1979-07-24 US disclosed
US-4136187-A CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DE) 1979-01-23 US disclosed
US-4004014-A VASODILATION, HYPOTENSIVE, ANTIARRHYTHMIA, SPASMOLYTIC BAYER AKTIENGESELLSCHAFT (DT) 1977-01-18 US disclosed
US-3959292-A HYPOTENSIVE AGENTS, CORONARY DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-05-25 US disclosed