SCHEMBL11565

SCHEMBL11565

O=C(Cc1ccc2ccccc2n1)N1CCNCC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.50
CYP3A4 P08684 3/20 0.49
KDM4E B2RXH2 3/20 0.49
HSD17B10 Q99714 2/20 0.49
ALDH1A1 P00352 3/20 0.49
HTR3E A5X5Y0 1/20 0.49
USP2 O75604 1/20 0.49
HTR3B O95264 1/20 0.49
ADRB1 P08588 1/20 0.49
HTR1A P08908 1/20 0.49
HTR2C P28335 1/20 0.49
MAPK1 P28482 1/20 0.49
SLC6A4 P31645 1/20 0.49
HTR7 P34969 1/20 0.49
HTT P42858 1/20 0.49
HTR3A P46098 1/20 0.49
HTR6 P50406 1/20 0.49
PMP22 Q01453 1/20 0.49
HTR3D Q70Z44 1/20 0.49
HTR3C Q8WXA8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1243996 0.75 KDM4E (0.59) KDM4EHSD17B10ALDH1A1SLC6A4SCN7A
SCHEMBL14198735 0.75 SLC6A4 (0.56) HTR3EHTR3BHTR2CSLC6A4HTR3A
SCHEMBL5139469 0.75 TSHR (0.66) CYP1A2CYP3A4KDM4EHSD17B10ALDH1A1
SCHEMBL3585730 0.75 POLB (0.55) CYP1A2CYP3A4KDM4EHSD17B10ALDH1A1
SCHEMBL29756443 0.75 CYP3A4 (0.55) CYP1A2CYP3A4KDM4EHSD17B10ALDH1A1
SCHEMBL2170401 0.75 CYP3A4 (0.55) CYP1A2CYP3A4KDM4EHSD17B10ALDH1A1
Hydrochloric Acid SCHEMBL6586965 0.74 TSHR (0.64) CYP1A2CYP3A4KDM4EHSD17B10ALDH1A1
SCHEMBL92506 0.74 L3MBTL1 (0.63) KDM4EALDH1A1USP2HTTLMNA
SCHEMBL3917010 0.74 CXCR4 (0.57) CYP1A2CYP3A4KDM4EHSD17B10ALDH1A1
SCHEMBL14805320 0.73 CYP1A2 (0.67) CYP1A2KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499144-A1 QUINOLINE AND QUINOXALINE DERIVATIVES AS KINASE INHIBITORS UCB Pharma, S.A. (BE) 2012-09-19 EP disclosed
WO-2011058110-A1 QUINOLINE AND QUINOXALINE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2011-05-19 WO disclosed