SCHEMBL11565858

SCHEMBL11565858

CCC(=O)C1(N(C(=O)C2CC2)c2ccccc2)CCN(CCc2ccccc2)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 14/20 0.61
OPRD1 P41143 6/20 0.61
OPRK1 P41145 3/20 0.61
SLC22A1 O15245 1/20 0.54
NR1I2 O75469 1/20 0.54
ABCB1 P08183 1/20 0.54
CHRM1 P11229 1/20 0.54
DRD2 P14416 1/20 0.54
ADRA2B P18089 1/20 0.54
ADRA2C P18825 1/20 0.54
CHRM3 P20309 1/20 0.54
MAOA P21397 1/20 0.54
DRD4 P21917 1/20 0.54
MAOB P27338 1/20 0.54
ADRA1A P35348 1/20 0.54
HRH1 P35367 1/20 0.54
ADRA1B P35368 1/20 0.54
DRD3 P35462 1/20 0.54
CHRNA4 P43681 1/20 0.54
SLC6A3 Q01959 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11563434 0.90 OPRM1 (0.60) OPRM1OPRD1OPRK1SLC22A1NR1I2
SCHEMBL11569033 0.88 OPRM1 (0.78) OPRM1OPRD1OPRK1
SCHEMBL11796741 0.87 OPRM1 (0.77) OPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL11567839 0.87 OPRM1 (0.69) OPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL11569081 0.86 OPRM1 (0.76) OPRM1OPRD1OPRK1
SCHEMBL9153525 0.83 OPRM1 (0.53) OPRM1OPRD1OPRK1SLC22A1NR1I2
Hydrochloric Acid SCHEMBL11565087 0.80 OPRM1 (0.76) OPRM1OPRD1OPRK1SLC22A1ABCB1
SCHEMBL3303683 0.80 OPRM1 (0.80) OPRM1OPRD1OPRK1
SCHEMBL11564033 0.79 OPRM1 (0.71) OPRM1OPRD1OPRK1
SCHEMBL821488 0.79 OPRM1 (0.78) OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4179569-A ANALGESIC INTERMEDIATES JANSSEN PHARMACEUTICA N.V. (BE) 1979-12-18 US disclosed
US-3998834-A ANALGESICS JANSSEN PHARMACEUTICA N.V. (BE) 1976-12-21 US disclosed