SCHEMBL11587716

SCHEMBL11587716

CCN(CC)S(=O)(=O)c1ccc2c(c1)C(CC(=O)O)c1ccccc1C(F)(F)C2(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.40
LMNA P02545 3/20 0.40
TSHR P16473 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 6/20 0.39
NPSR1 Q6W5P4 2/20 0.39
MAPT P10636 2/20 0.39
HTT P42858 2/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C9 P11712 2/20 0.39
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11587097 0.86 CYP2C9 (0.39) TSHRMEN1KMT2AALDH1A1KDM4E
SCHEMBL11585751 0.83 ALDH1A1 (0.39) SMN1; SMN2LMNATSHRMEN1KMT2A
SCHEMBL11586952 0.83 ALDH1A1 (0.46) SMN1; SMN2LMNATSHRMEN1KMT2A
SCHEMBL11632020 0.83 ALDH1A1 (0.43) SMN1; SMN2LMNATSHRMEN1KMT2A
SCHEMBL11588145 0.81 ALDH1A1 (0.43) SMN1; SMN2LMNATSHRALDH1A1NPSR1
SCHEMBL11882597 0.79 HTT (0.38) SMN1; SMN2LMNATSHRALDH1A1NPSR1
SCHEMBL11587148 0.78 EGFR (0.49) TSHRMAPTCYP1A2
SCHEMBL11587254 0.78 EGFR (0.40) SMN1; SMN2LMNAMAPT
SCHEMBL11587935 0.77 ALDH1A1 (0.40) SMN1; SMN2LMNATSHRKMT2AALDH1A1
SCHEMBL11585500 0.75 EGFR (0.40) MEN1KMT2AMAPTCYP2C9PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4070387-A ANTIARRHYTHMIC AGENTS MERCK & CO., INC. (US) 1978-01-24 US disclosed
US-4020096-A ANTIARRYTHMIA MERCK & CO., INC. (US) 1977-04-26 US disclosed
US-3950423-A 10,11-Dihydro-10,10,11,11-tetrafluoro-5H-dibenzo[a,d]cycloheptene-5-methylamines MERCK & CO., INC. (US) 1976-04-13 US disclosed