SCHEMBL11596065

SCHEMBL11596065

Cc1cc2n(C)c(=O)c3cnccc3n2n1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
PDE10A Q9Y233 2/20 0.41
TOP2A P11388 1/20 0.38
CYP1A2 P05177 1/20 0.37
PARP1 P09874 1/20 0.37
GRM4 Q14833 1/20 0.36
ELANE P08246 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11622420 0.89 TOP2A (0.41) KDM4EALDH1A1PDE10ATOP2ACYP1A2
SCHEMBL11595420 0.76 KDM4E (0.38) KDM4EALDH1A1CYP1A2PARP1
SCHEMBL11595529 0.74 KDM4E (0.34) KDM4EALDH1A1
SCHEMBL31256305 0.72 TOP2A (0.50) KDM4EPDE10ATOP2A
SCHEMBL17627450 0.72 TOP2A (0.40) KDM4EALDH1A1TOP2A
SCHEMBL11598229 0.72 KDM4E (0.36) KDM4EALDH1A1
SCHEMBL9534299 0.72 ADORA3 (0.49) KDM4EALDH1A1CYP1A2GRM4CYP2D6
SCHEMBL11596500 0.71 PARP1 (0.68) KDM4EALDH1A1CYP1A2PARP1
SCHEMBL22845397 0.69 KDM4E (0.43) KDM4EALDH1A1CYP1A2
SCHEMBL17627424 0.69 KDM4E (0.38) KDM4EALDH1A1TOP2AGRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4066645-A Derivatives of pyrazolo [1,5-a]pyrido[3,4-e]pyrimidine E. R. SQUIBB & SONS, INC. (US) 1978-01-03 US disclosed